Uniprot accession / id : P10275  OR   Uniprot accession / id : Q9TT90  OR   Uniprot accession / id : B1AVE7  OR   Uniprot accession / id : P19091  OR   Uniprot accession / id : P15207  OR   Uniprot accession / id : Q2ACE0
 
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Entry Information
Entry status  (1)
REL
(103)
 
Experimental methods  (1)
X-ray diffraction
(103)
 
Authors  (371)
Estebanez-Perpina E
(21)
Estébanez-Perpiñá E
(21)
Hsu CL
(21)
Liu JS
(21)
Wu WG
(21)
Chang C
(20)
Chen CJ
(20)
Chen YL
(20)
Guan HH
(20)
Guy RK
(20)
Lin AC
(20)
Ma WL
(20)
Pang ST
(20)
Ting HJ
(20)
Wu PL
(20)
Yeh SD
(20)
Fletterick RJ
(16)
Baxter JD
(15)
Mar E
(15)
Nguyen P
(15)
Webb P
(15)
Bohl CE
(14)
Dalton JT
(14)
Miller DD
(14)
Arnold LA
(12)
Bell CE
(12)
Arnold AA
(11)
Bateman R
(11)
Pallai P
(11)
Rodrigues ED
(11)
Shokat KM
(11)
Chen J
(10)
Fletterick KR
(9)
Cherkasov A
(7)
Gampe RT
(7)
Leblanc E
(7)
Rennie PS
(7)
Stanley TB
(7)
Wilson EM
(7)
Abella M
(6)
An Y
(6)
Axerio-Cilies P
(6)
Fuentes-Prior P
(6)
Krystek SR
(6)
Lack NA
(6)
LeBlanc E
(6)
Wu Z
(6)
Alegre-Marti A
(5)
Alegre-Martí A
(5)
Anton R
(5)
Antón R
(5)
Aytes A
(5)
Aytes Á
(5)
Chan KH
(5)
Chinas M
(5)
Chiñas M
(5)
Doamekpor SK
(5)
Eckhard U
(5)
Fernandez-Recio J
(5)
Fernández-Recio J
(5)
Han FQ
(5)
Hwang DJ
(5)
Jimenez-Panizo A
(5)
Jiménez-Panizo A
(5)
Le Romancer M
(5)
Ma L
(5)
Martinez-Tebar A
(5)
Martínez-Tébar A
(5)
Mohler ML
(5)
Mustafa S
(5)
Peng P
(5)
Peralta-Moreno MN
(5)
Piulats JM
(5)
Poulard C
(5)
Rojas AM
(5)
Rubio-Martinez J
(5)
Rubio-Martínez J
(5)
Sack JS
(5)
Tong L
(5)
Tong Y
(5)
Xu R
(5)
Yang J
(5)
Askew EB
(4)
Axerio P
(4)
Breton R
(4)
Buehrer BM
(4)
Cantin L
(4)
Claessens F
(4)
Delgado-Rodrigues E
(4)
Faggart JL
(4)
Feau C
(4)
Guns ET
(4)
Kish KF
(4)
Kuchenbecker K
(4)
Labrie F
(4)
Moore JM
(4)
Moore JMR
(4)
Pereira de Jesus-Tran K
(4)
Salvati ME
(4)
Tavassoli P
(4)
 
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Homo / hetero assembly  (2)
homo
(63)
hetero
(40)
 
Assembly composition  (3)
protein structure
(63)
protein/protein complex
(37)
DNA/protein complex
(3)
 
Assembly polymer count  (4)
monomer
(63)
dimer
(36)
tetramer
(3)
hexamer
(1)
 
Resolution distribution
1.0 - 1.5
(5)
1.5 - 2
(49)
2.0 - 2.5
(33)
2.5 - 3
(12)
3.0 - 3.5
(3)
3.5 - 4
(1)
 
Representative Structures
Representative Structures
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Entries 1 to 10 of 103
Entries 1 to 10 of 103
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Crystal structure of mutant Androgen Receptor ligand binding domain F877L/T878A with DHT
Doamekpor SK, Tong L
Acta Crystallogr F Struct Biol Commun (2023) [PMID: 36995121  ]
Source organism: Homo sapiens  
Assembly composition: protein only structure
Bound ligands: DHT    SO4    DHT   
Assembly name: Androgen receptor (Preferred)   search this complex
PDBe complex ID: PDB-CPX-145222 (Preferred)   search this ID
PDBe-KB: P10275   
X-ray diffraction
1.69Å resolution
Released: 12 Apr 2023
Model geometry
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8fh1
8fh1
8fh1
Crystal Structure of Human Androgen Receptor DNA Binding Domain Bound to its Response Element: C3(1)ARE
Lee XY, Helsen C, Van Eynde W, Voet A, Claessens F
J Steroid Biochem Mol Biol (2024) [PMID: 38604378  ]
Source organism: Homo sapiens  
Assembly composition: DNA/protein complex
Bound ligands: ZN    ZN   
Assembly name: Androgen receptor and DNA (Preferred)   search this complex
PDBe complex ID: PDB-CPX-270706 (Preferred)   search this ID
PDBe-KB: P10275   
X-ray diffraction
2.05Å resolution
Released: 24 Apr 2024
Model geometry
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8rm6
8rm6
8rm6
Crystal structure of mutant Androgen Receptor ligand binding domain L702H/H875Y/F877L with DHT
Doamekpor SK, Tong L
Acta Crystallogr F Struct Biol Commun (2023) [PMID: 36995121  ]
Source organism: Homo sapiens  
Assembly composition: protein only structure
Bound ligands: DHT    SO4    DHT   
Assembly name: Androgen receptor (Preferred)   search this complex
PDBe complex ID: PDB-CPX-145222 (Preferred)   search this ID
PDBe-KB: P10275   
X-ray diffraction
1.61Å resolution
Released: 12 Apr 2023
Model geometry
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8fgz
8fgz
8fgz
Crystal structure of mutant Androgen Receptor ligand binding domain L702H/H875Y with DHT
Doamekpor SK, Tong L
Acta Crystallogr F Struct Biol Commun (2023) [PMID: 36995121  ]
Source organism: Homo sapiens  
Assembly composition: protein only structure
Bound ligands: DHT    SO4    DHT   
Assembly name: Androgen receptor (Preferred)   search this complex
PDBe complex ID: PDB-CPX-145222 (Preferred)   search this ID
PDBe-KB: P10275   
X-ray diffraction
1.59Å resolution
Released: 12 Apr 2023
Model geometry
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8fh2
8fh2
8fh2
Crystal structure of mutant Androgen Receptor ligand binding domain L702H/H875Y/F877L/T878A with DHT
Doamekpor SK, Tong L
Acta Crystallogr F Struct Biol Commun (2023) [PMID: 36995121  ]
Source organism: Homo sapiens  
Assembly composition: protein only structure
Bound ligands: DHT    DHT   
Assembly name: Androgen receptor (Preferred)   search this complex
PDBe complex ID: PDB-CPX-145222 (Preferred)   search this ID
PDBe-KB: P10275   
X-ray diffraction
2.2Å resolution
Released: 12 Apr 2023
Model geometry
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8fgy
8fgy
8fgy
Crystal Structure of Homodimeric Androgen Receptor Ligand-Binding Domain bound to DHT and LxxLL peptide
Estebanez-Perpina E, Fuentes-Prior P
Nat Commun (2017) [PMID: 28165461  ]
Source organism: Homo sapiens  
Assembly composition: protein/protein complex
Bound ligands: ACT    GOL    ZN    DHT    SO4    ZN    CL    EDO    ACT    DHT    PGE    PGE   
Modified residues: FME    SNC    FME    SNC   
PDBe complex ID: PDB-CPX-145224 (Preferred)   search this ID
PDBe-KB: P10275    Q8TBC4   
X-ray diffraction
2.15Å resolution
Released: 15 Mar 2017
Model geometry
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5jjm
5jjm
5jjm
Synthesis and biological evaluation of novel selective androgen receptor modulators (SARMs): Part III
Wilson KP
Bioorg Med Chem (2017) [PMID: 28454849  ]
Source organism: Homo sapiens  
Assembly composition: protein only structure
Bound ligands: GOL    97A    97A   
Assembly name: Androgen receptor (Preferred)   search this complex
PDBe complex ID: PDB-CPX-145222 (Preferred)   search this ID
PDBe-KB: P10275   
X-ray diffraction
1.44Å resolution
Released: 24 May 2017
Model geometry
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5v8q
5v8q
5v8q
Crystal Structure of a Selective Androgen Receptor Modulator Bound to the Ligand Binding Domain of the Human Androgen Receptor
Luz JG, Saeed A, Wang Y
J Med Chem (2016) [PMID: 26683992  ]
Assembly composition: protein/protein complex
Bound ligands: 51Y    51Y   
Assembly name: Androgen receptor (Preferred)   search this complex
PDBe complex ID: PDB-CPX-145223 (Preferred)   search this ID
PDBe-KB: P10275   
X-ray diffraction
2.07Å resolution
Released: 6 Jan 2016
Model geometry
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5cj6
5cj6
5cj6
Crystal Structure Of The Androgen Receptor Ligand Binding Domain In Complex With 5-(2-fluoro-4-hydroxyphenyl)-1-methyl-1H-pyrrole-2-carbonitrile
Parris K, Unwalla R
J Med Chem (2017) [PMID: 28696695  ]
Source organism: Homo sapiens  
Assembly composition: protein only structure
Bound ligands: 9FG    9FG   
Assembly name: Androgen receptor (Preferred)   search this complex
PDBe complex ID: PDB-CPX-145222 (Preferred)   search this ID
PDBe-KB: P10275   
X-ray diffraction
2.35Å resolution
Released: 14 Mar 2018
Model geometry
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5vo4
5vo4
5vo4
Synthesis and biological evaluation of novel selective androgen receptor modulators (SARMs). Part II: Optimization of 4-(pyrrolidin-1-yl)benzonitrile derivatives
Wilson KP
Bioorg Med Chem Lett (2017) [PMID: 28363748  ]
Source organism: Homo sapiens  
Assembly composition: protein only structure
Bound ligands: 77U    GOL    77U   
Assembly name: Androgen receptor (Preferred)   search this complex
PDBe complex ID: PDB-CPX-145222 (Preferred)   search this ID
PDBe-KB: P10275   
X-ray diffraction
2.71Å resolution
Released: 26 Apr 2017
Model geometry
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5t8e
5t8e
5t8e
...
Entries 1 to 10 of 103
Entries 1 to 10 of 103