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Showing 1-20 out of 22 records

#	Molecule ChEMBL ID	Compound Key	Standard Type	Standard Relation	Standard Value	Standard Text Value	Standard Units	pChEMBL Value	Comment	Assay ChEMBL ID	Assay Description	BAO Label	Assay Organism	Target ChEMBL ID	Target Name	Target Organism	Target Type	Document ChEMBL ID	Source Description	Cell ChEMBL ID
1.	Error: . CHEMBL204785	2	CL	=	11.0	---	mL.min-1.kg-1	---	---	CHEMBL912127	Clearance in Wistar rat at 3 mg/kg, iv	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1149524	Scientific Literature	---
2.	Error: . CHEMBL204785	3	F	<	1.0	---	%	---	---	CHEMBL863810	Oral bioavailability in Wistar rat at 10 mg/kg, po	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1146936	Scientific Literature	---
3.	Error: . CHEMBL204785	3	Ki	=	29.0	---	nM	7.54	---	CHEMBL863796	Inhibition of Cathepsin S	single protein format	Homo sapiens	CHEMBL2954	Cathepsin S	Homo sapiens	SINGLE PROTEIN	CHEMBL1146936	Scientific Literature	---
4.	Error: . CHEMBL204785	3	Vdss	=	1.63	---	L.kg-1	---	---	CHEMBL863805	Volume of distribution in Wistar rat at 3 mg/kg, iv	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1146936	Scientific Literature	---
5.	Error: . CHEMBL204785	3	T1/2	=	4.8	---	hr	---	---	CHEMBL863806	Half life in Wistar rat at 3 mg/kg, iv	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1146936	Scientific Literature	---
6.	Error: . CHEMBL204785	2	Stability	=	4.0	---	%	---	---	CHEMBL912125	Stability in rat liver microsomes	microsome format	Rattus norvegicus	CHEMBL613694	Liver microsomes	Rattus norvegicus	SUBCELLULAR	CHEMBL1149524	Scientific Literature	---
7.	Error: . CHEMBL204785	3	Ki	>	10000.0	---	nM	---	---	CHEMBL863798	Inhibition of Cathepsin L	single protein format	Homo sapiens	CHEMBL3837	Cathepsin L	Homo sapiens	SINGLE PROTEIN	CHEMBL1146936	Scientific Literature	---
8.	Error: . CHEMBL204785	3	Ki	>	100000.0	---	nM	---	---	CHEMBL863799	Inhibition of Cathepsin B	single protein format	Homo sapiens	CHEMBL4072	Cathepsin B	Homo sapiens	SINGLE PROTEIN	CHEMBL1146936	Scientific Literature	---
9.	Error: . CHEMBL204785	2	Solubility	=	10.0	---	ug.mL-1	---	---	CHEMBL912124	Solubility at pH 6.8	small-molecule physicochemical format	---	CHEMBL2362975	No relevant target	---	NO TARGET	CHEMBL1149524	Scientific Literature	---
10.	Error: . CHEMBL204785	3	AUC	=	15.0	---	ng.hr.mL-1	---	---	CHEMBL863807	AUC in Wistar rat at 10 mg/kg, po	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1146936	Scientific Literature	---
11.	Error: . CHEMBL204785	3	Ki	>	30000.0	---	nM	---	---	CHEMBL863797	Inhibition of Cathepsin K	single protein format	Homo sapiens	CHEMBL268	Cathepsin K	Homo sapiens	SINGLE PROTEIN	CHEMBL1146936	Scientific Literature	---
12.	Error: . CHEMBL204785	2	Cmax	=	12.0	---	nM	---	---	CHEMBL912130	Cmax in Wistar rat at 10 mg/kg, po	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1149524	Scientific Literature	---
13.	Error: . CHEMBL204785	2	Vdss	=	1.63	---	L.kg-1	---	---	CHEMBL912128	Volume of distribution in Wistar rat at 3 mg/kg, iv	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1149524	Scientific Literature	---
14.	Error: . CHEMBL204785	3	Cp	---	---	---	---	---	Not Active	CHEMBL863802	Plasma concentration in Wistar rat at 10 mg/kg, po	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1146936	Scientific Literature	---
15.	Error: . CHEMBL204785	3	CL	=	11.4	---	mL.min-1.kg-1	---	---	CHEMBL863804	Clearance in Wistar rat at 3 mg/kg, iv	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1146936	Scientific Literature	---
16.	Error: . CHEMBL204785	2	F	<	1.0	---	%	---	---	CHEMBL912132	Bioavailability in Wistar rat at 10 mg/kg, po	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1149524	Scientific Literature	---
17.	Error: . CHEMBL204785	2	T1/2	=	4.8	---	hr	---	---	CHEMBL912126	Half life in Wistar rat at 3 mg/kg, iv	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1149524	Scientific Literature	---
18.	Error: . CHEMBL204785	2	AUC	=	15.0	---	ng.hr.mL-1	---	---	CHEMBL912131	AUC in Wistar rat at 10 mg/kg, po	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1149524	Scientific Literature	---
19.	Error: . CHEMBL204785	2	T1/2	=	5.3	---	hr	---	---	CHEMBL912129	Half life in Wistar rat at 10 mg/kg, po	organism-based format	Rattus norvegicus	CHEMBL376	Rattus norvegicus	Rattus norvegicus	ORGANISM	CHEMBL1149524	Scientific Literature	---
20.	Error: . CHEMBL204785	3	Stability	<	5.0	---	%	---	---	CHEMBL863803	Metabolic stability in Wistar rat liver microsome	microsome format	Rattus norvegicus	CHEMBL613694	Liver microsomes	Rattus norvegicus	SUBCELLULAR	CHEMBL1146936	Scientific Literature	---

Showing 1-20 out of 22 records

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