Activities
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| # | Molecule ChEMBL ID | Compound Key | Standard Type | Standard Relation | Standard Value | Standard Text Value | Standard Units | pChEMBL Value | Comment | Assay ChEMBL ID | Assay Description | BAO Label | Assay Organism | Target ChEMBL ID | Target Name | Target Organism | Target Type | Document ChEMBL ID | Source Description | Cell ChEMBL ID | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |
SID103905260
|
Ki
|
>
|
5011.87
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: INSR
|
assay format
|
---
|
Insulin receptor
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 2. |
SID103905260
|
Ki
|
=
|
63.1
|
---
|
nM
|
7.20
|
active
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: PLK4
|
assay format
|
---
|
Serine/threonine-protein kinase PLK4
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 3. |
SID103905260
|
Ki
|
=
|
39.81
|
---
|
nM
|
7.40
|
active
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: PRKD2
|
assay format
|
---
|
Serine/threonine-protein kinase D2
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 4. |
SID103905260
|
Ki
|
>
|
1584.89
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: PRKG2
|
assay format
|
---
|
cGMP-dependent protein kinase 2
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 5. |
SID103905260
|
Ki
|
>
|
1995.26
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: FES
|
assay format
|
---
|
Tyrosine-protein kinase FES
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 6. |
SID103905260
|
Ki
|
>
|
1995.26
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: MATK
|
assay format
|
---
|
Tyrosine-protein kinase CTK
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 7. |
SID103905260
|
Ki
|
>
|
7943.28
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: MAPK13
|
assay format
|
---
|
MAP kinase p38 delta
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 8. |
16
|
IC50
|
=
|
81.0
|
---
|
nM
|
7.09
|
---
|
Inhibition of MK5
|
single protein format
|
Homo sapiens
|
MAP kinase-activated protein kinase 5
|
Homo sapiens
|
SINGLE PROTEIN
|
Scientific Literature
| ||||||
| 9. |
16
|
IC50
|
=
|
5700.0
|
---
|
nM
|
5.24
|
---
|
Inhibition of MNK1
|
single protein format
|
Homo sapiens
|
MAP kinase-interacting serine/threonine-protein kinase MNK1
|
Homo sapiens
|
SINGLE PROTEIN
|
Scientific Literature
| ||||||
| 10. |
SID103905260
|
Ki
|
>
|
1995.26
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: FGFR3
|
assay format
|
---
|
Fibroblast growth factor receptor 3
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 11. |
SID103905260
|
Ki
|
=
|
1000.0
|
---
|
nM
|
6.00
|
active
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: PRKAA1
|
assay format
|
---
|
AMP-activated protein kinase, alpha-1 subunit
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 12. |
SID103905260
|
Ki
|
=
|
25.12
|
---
|
nM
|
7.60
|
active
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: DAPK3
|
assay format
|
---
|
Death-associated protein kinase 3
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 13. |
SID103905260
|
Ki
|
>
|
1258.93
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: MELK
|
assay format
|
---
|
Maternal embryonic leucine zipper kinase
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 14. |
SID103905260
|
Ki
|
=
|
79.43
|
---
|
nM
|
7.10
|
active
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: DYRK3
|
assay format
|
---
|
Dual-specificity tyrosine-phosphorylation regulated kinase 3
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 15. |
SID103905260
|
Ki
|
>
|
1584.89
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: IGF1R
|
assay format
|
---
|
Insulin-like growth factor I receptor
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 16. |
SID103905260
|
Ki
|
=
|
316.23
|
---
|
nM
|
6.50
|
active
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: DYRK4
|
assay format
|
---
|
Dual specificity tyrosine-phosphorylation-regulated kinase 4
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 17. |
SID103905260
|
Ki
|
>
|
10000.0
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: LIMK1
|
assay format
|
---
|
LIM domain kinase 1
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 18. |
SID103905260
|
Ki
|
=
|
3981.07
|
---
|
nM
|
5.40
|
active
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: CAMK2G
|
assay format
|
---
|
CaM kinase II gamma
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 19. |
SID103905260
|
Ki
|
>
|
1584.89
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: LYN
|
assay format
|
---
|
Tyrosine-protein kinase Lyn
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
| ||||||
| 20. |
SID103905260
|
Ki
|
>
|
3162.28
|
---
|
nM
|
---
|
inactive
|
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: IKBKB
|
assay format
|
---
|
Inhibitor of nuclear factor kappa B kinase beta subunit
|
Homo sapiens
|
SINGLE PROTEIN
|
PubChem BioAssays
|
Showing 1-20
out of 163 records
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