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Showing 1-20 out of 115 records

#	Molecule ChEMBL ID	Compound Key	Standard Type	Standard Relation	Standard Value	Standard Text Value	Standard Units	pChEMBL Value	Comment	Assay ChEMBL ID	Assay Description	BAO Label	Assay Organism	Target ChEMBL ID	Target Name	Target Organism	Target Type	Document ChEMBL ID	Source Description	Cell ChEMBL ID
1.	Error: . CHEMBL292303	8	KA	=	41.0	---	uM	---	---	CHEMBL1067708	Activation of human recombinant CA1 by stopped flow CO2 hydration assay	single protein format	Homo sapiens	CHEMBL261	Carbonic anhydrase I	Homo sapiens	SINGLE PROTEIN	CHEMBL1157628	Scientific Literature	---
2.	Error: . CHEMBL292303	8	KA	=	41.0	---	uM	---	---	CHEMBL4233789	Activation of human CA1 by stopped-flow CO2 hydration assay	single protein format	Homo sapiens	CHEMBL261	Carbonic anhydrase I	Homo sapiens	SINGLE PROTEIN	CHEMBL4229443	Scientific Literature	---
3.	Error: . CHEMBL292303	8	KA	=	19.0	---	uM	---	---	CHEMBL1067711	Activation of Stylophora pistillata carbonic anhydrase STPCA by stopped flow CO2 hydration assay	assay format	Stylophora pistillata	CHEMBL612545	Unchecked	---	UNCHECKED	CHEMBL1157628	Scientific Literature	---
4.	Error: . CHEMBL292303	8	KA	=	33.0	---	uM	---	---	CHEMBL3870985	Activation of recombinant Methanosarcina thermophila gamma carbonic anhydrase at 10 uM incubated for 15 mins prior to testing by stopped flow CO2 hydration assay	single protein format	Methanosarcina thermophila	CHEMBL3932	Carbonic anhydrase	Methanosarcina thermophila	SINGLE PROTEIN	CHEMBL3870339	Scientific Literature	---
5.	Error: . CHEMBL292303	8, D-Trp	KA	=	0.002	---	uM	---	---	CHEMBL2156562	Activity of Sulfurihydrogenibium yellowstonense YO3AOP1 recombinant CA expressed in Escherichia coli BL21(DE3) after 15 mins by phenol red staining based stopped flow CO2 hydration assay	assay format	Sulfurihydrogenibium yellowstonense	CHEMBL612545	Unchecked	---	UNCHECKED	CHEMBL2150956	Scientific Literature	---
6.	Error: . CHEMBL292303	D-Trp	Ka	=	18.0	---	uM	---	---	CHEMBL987042	Activation of human recombinant CA14 after 15 mins by stopped-flow CO2 hydration assay	single protein format	Homo sapiens	CHEMBL3510	Carbonic anhydrase XIV	Homo sapiens	SINGLE PROTEIN	CHEMBL1144196	Scientific Literature	---
7.	Error: . CHEMBL292303	SID144204756	Potency	---	19952.6	---	nM	---	inconclusive	CHEMBL3214970	PubChem BioAssay. qHTS Assay for Identifying Gametocytocidal Compounds. (Class of assay: confirmatory)	assay format	---	CHEMBL612545	Unchecked	---	UNCHECKED	CHEMBL1201862	PubChem BioAssays	---
8.	Error: . CHEMBL292303	8, D-Trp	Ka	=	19.0	---	uM	---	---	CHEMBL970752	Activation of human recombinant CA3 at 10 uM by stopped-flow CO2 hydration method	single protein format	Homo sapiens	CHEMBL2885	Carbonic anhydrase III	Homo sapiens	SINGLE PROTEIN	CHEMBL1155874	Scientific Literature	---
9.	Error: . CHEMBL292303	8, D-Trp	KA	=	41.0	---	uM	---	---	CHEMBL932481	Activation of human recombinant CA1 by stopped-flow CO2 hydration method	single protein format	Homo sapiens	CHEMBL261	Carbonic anhydrase I	Homo sapiens	SINGLE PROTEIN	CHEMBL1142388	Scientific Literature	---
10.	Error: . CHEMBL292303	D-tryptophan	Ki	=	880000.0	---	nM	---	---	CHEMBL4621660	Inhibition of human DHFR in presence of DHF and NADPH by UV-vis spectrometry by Lineweaver-Burk plot analysis	single protein format	Homo sapiens	CHEMBL202	Dihydrofolate reductase	Homo sapiens	SINGLE PROTEIN	CHEMBL4619782	Scientific Literature	---
11.	Error: . CHEMBL292303	8	KA	=	12.0	---	uM	---	---	CHEMBL4233790	Activation of human CA2 by stopped-flow CO2 hydration assay	single protein format	Homo sapiens	CHEMBL205	Carbonic anhydrase II	Homo sapiens	SINGLE PROTEIN	CHEMBL4229443	Scientific Literature	---
12.	Error: . CHEMBL292303	SID170465485	Ac50	---	0.7943	---	uM	---	inactive	CHEMBL3561990	PubChem BioAssay. qHTS Assay for Identifying Compounds that block Entry of Ebola Virus: Screen 2, green channel. (Class of assay: confirmatory)	assay format	---	CHEMBL612545	Unchecked	---	UNCHECKED	CHEMBL1201862	PubChem BioAssays	---
13.	Error: . CHEMBL292303	10	KA	=	1.3	---	uM	---	---	CHEMBL5037979	Activation of human carbonic anhydrase 5B by stopped flow assay	single protein format	Homo sapiens	CHEMBL3969	Carbonic anhydrase VB	Homo sapiens	SINGLE PROTEIN	CHEMBL5036350	Scientific Literature	---
14.	Error: . CHEMBL292303	8	Ka	=	28.0	---	uM	---	---	CHEMBL987040	Activation of human recombinant CA12 after 15 mins by stopped-flow CO2 hydration assay	single protein format	Homo sapiens	CHEMBL3242	Carbonic anhydrase XII	Homo sapiens	SINGLE PROTEIN	CHEMBL1144196	Scientific Literature	---
15.	Error: . CHEMBL292303	D-Tryptophan	Activity	---	---	---	---	---	is not an inhibitor [-]	CHEMBL2076200	TP_TRANSPORTER: inhibition of L-tryptophan uptake in Xenopus laevis oocytes	cell-based format	Xenopus laevis	CHEMBL2073717	Monocarboxylate transporter 10	Rattus norvegicus	SINGLE PROTEIN	CHEMBL2074257	TP-search Transporter Database	CHEMBL3308859
16.	Error: . CHEMBL292303	D-Trp	KA	=	12.0	---	uM	---	---	CHEMBL1067709	Activation of human recombinant CA2by stopped flow CO2 hydration assay	single protein format	Homo sapiens	CHEMBL205	Carbonic anhydrase II	Homo sapiens	SINGLE PROTEIN	CHEMBL1157628	Scientific Literature	---
17.	Error: . CHEMBL292303	D-Trp	Kcat	=	6.1	---	10'5/s	---	---	CHEMBL1067705	Activity of human recombinant CA2at 10 uM by stopped flow CO2 hydration assay	single protein format	Homo sapiens	CHEMBL205	Carbonic anhydrase II	Homo sapiens	SINGLE PROTEIN	CHEMBL1157628	Scientific Literature	---
18.	Error: . CHEMBL292303	D-Trp	Kcat	=	4.8	---	10'5/s	---	---	CHEMBL1067706	Activity of human full length CA6 at 10 uM by stopped flow CO2 hydration assay	single protein format	Homo sapiens	CHEMBL3025	Carbonic anhydrase VI	Homo sapiens	SINGLE PROTEIN	CHEMBL1157628	Scientific Literature	---
19.	Error: . CHEMBL292303	D-Trp	Kcat	=	6.4	---	10'5/s	---	---	CHEMBL1067707	Activity of Stylophora pistillata carbonic anhydrase STPCA at 10 uM by stopped flow CO2 hydration assay	assay format	Stylophora pistillata	CHEMBL612545	Unchecked	---	UNCHECKED	CHEMBL1157628	Scientific Literature	---
20.	Error: . CHEMBL292303	SID26753353	Potency	---	33498.3	---	nM	---	inconclusive	CHEMBL2114780	PubChem BioAssay. A quantitative high throughput screen for small molecules that induce DNA re-replication in SW480 colon adenocarcinoma cells. (Class of assay: confirmatory)	cell-based format	Homo sapiens	CHEMBL1293278	Geminin	Homo sapiens	SINGLE PROTEIN	CHEMBL1201862	PubChem BioAssays	CHEMBL3307758

Showing 1-20 out of 115 records

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