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Showing 1-14 out of 14 records

	#	Molecule ChEMBL ID	Compound Key	Standard Type	Standard Relation	Standard Value	Standard Text Value	Standard Units	pChEMBL Value	Comment	Assay ChEMBL ID	Assay Description	BAO Label	Assay Organism	Target ChEMBL ID	Target Name	Target Organism	Target Type	Document ChEMBL ID	Source Description	Cell ChEMBL ID
	1.	Error: . CHEMBL993	Thymine	EC90	---	---	---	---	---	Not Determined	CHEMBL763513	The anti-HIV-1 activity was assayed in activated human peripheral blood mononuclear (PBM) cells, relative to RVT; not determined	assay format	Homo sapiens	CHEMBL612558	ADMET	---	ADMET	CHEMBL1137958	Scientific Literature	---
	2.	Error: . CHEMBL993	4	Activity	---	---	---	---	---	Not Active	CHEMBL3280588	Antitumor activity against rat Walker 256 cells allografted in Sprague-Dawley rat at 2.5 mg/kg/day, ip relative to control	organism-based format	Rattus norvegicus	CHEMBL612803	W256	Rattus norvegicus	CELL-LINE	CHEMBL3271954	Scientific Literature	CHEMBL3307248
	3.	Error: . CHEMBL993	2	Ki	=	347000000.0	---	nM	---	---	CHEMBL815505	Inhibitory activity against mouse liver thymidine phosphorylase at 0.15 mM thymidine substrate	assay format	---	CHEMBL2606	Thymidine phosphorylase	Mus musculus	SINGLE PROTEIN	CHEMBL1136315	Scientific Literature	---
	4.	Error: . CHEMBL993	Thymine	EC50	---	---	---	nM	---	Not Determined	CHEMBL758447	The anti-HIV-1 activity was assayed in activated human peripheral blood mononuclear (PBM) cells, relative to RVT; not determined	assay format	Homo sapiens	CHEMBL612558	ADMET	---	ADMET	CHEMBL1137958	Scientific Literature	---
	5.	Error: . CHEMBL993	thymine	Activity	---	---	---	---	---	Not Active	CHEMBL1107320	Cytotoxicity against human KB cells at 30 uM	cell-based format	Homo sapiens	CHEMBL398	KB	Homo sapiens	CELL-LINE	CHEMBL1157067	Scientific Literature	CHEMBL3307959
	6.	Error: . CHEMBL993	Thymine	Kd	=	10000000.0	---	nM	2.00	---	CHEMBL3626885	Binding affinity to recombinant human ATAD2 (982 to 1108 amino acids) bromodomain radiolabelled at methyl groups of leucine, valine, isoleucine, methionine expressed in Escherichia coli BL21 (DE3) by NMR titration	assay format	Homo sapiens	CHEMBL2150837	ATPase family AAA domain-containing protein 2	Homo sapiens	SINGLE PROTEIN	CHEMBL3621199	Scientific Literature	---
	7.	Error: . CHEMBL993	Thymine	IC50	>	100000.0	---	nM	---	---	CHEMBL757722	Cytotoxicity was determined in PBM cells, relative to RVT	cell-based format	Homo sapiens	CHEMBL612558	ADMET	---	ADMET	CHEMBL1137958	Scientific Literature	---
	8.	Error: . CHEMBL993	Thymine	IC50	>	100000.0	---	nM	---	---	CHEMBL656431	Cytotoxicity was determined in CEM cells, relative to RVT	cell-based format	Homo sapiens	CHEMBL382	CCRF-CEM	Homo sapiens	CELL-LINE	CHEMBL1137958	Scientific Literature	CHEMBL3307641
	9.	Error: . CHEMBL993	18a	IC50	>	100.0	---	ug.mL-1	---	---	CHEMBL1227838	Cytotoxicity against MDCK cells	cell-based format	Canis lupus familiaris	CHEMBL614068	MDCK	Canis lupus familiaris	CELL-LINE	CHEMBL1221294	Scientific Literature	CHEMBL3308370
	10.	Error: . CHEMBL993	4	Activity	---	---	---	---	---	Not Active	CHEMBL3280589	Antitumor activity against mouse P388 cells allografted in DBA/2 mouse at 25 mg/kg/day, ip administered for 2 weeks relative to control	organism-based format	Mus musculus	CHEMBL389	P388	Mus musculus	CELL-LINE	CHEMBL3271954	Scientific Literature	CHEMBL3308401
	11.	Error: . CHEMBL993	4	Activity	---	---	---	---	---	Not Active	CHEMBL3280590	Antitumor activity against mouse B16 cells allografted in C57Bl/6 mouse at 25 mg/kg/day, ip administered for 2 weeks relative to control	organism-based format	Mus musculus	CHEMBL381	B16	Mus musculus	CELL-LINE	CHEMBL3271954	Scientific Literature	CHEMBL3308454
	12.	Error: . CHEMBL993	Thymine	IC50	>	100000.0	---	nM	---	---	CHEMBL818228	Cytotoxicity was determined in Vero cells, relative to RVT	cell-based format	Chlorocebus sabaeus	CHEMBL391	Vero	Chlorocebus sabaeus	CELL-LINE	CHEMBL1137958	Scientific Literature	CHEMBL3307520
	13.	Error: . CHEMBL993	18a	EC50	>	100.0	---	ug.mL-1	---	---	CHEMBL1227836	Antiviral activity against Influenza A virus H5N1 Vietnam/1203/2004H infected in MDCK cells	organism-based format	Influenza A virus	CHEMBL613740	Influenza A virus	Influenza A virus	ORGANISM	CHEMBL1221294	Scientific Literature	CHEMBL3308370
	14.	Error: . CHEMBL993	18a	EC50	>	100.0	---	ug.mL-1	---	---	CHEMBL1227837	Antiviral activity against Influenza B virus Florida/4/2006 infected in MDCK cells	cell-based format	Influenza B virus	CHEMBL613129	Influenza B virus	Influenza B virus	ORGANISM	CHEMBL1221294	Scientific Literature	CHEMBL3308370

Showing 1-14 out of 14 records

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