CryoEM structure of NaDC1 with Citrate
Resolution: 2.7 Å
EM Method: Single-particle
Fitted PDBs: 8w6c
Q-score: 0.631
Chi X, Chen Y, Li Y, Dai L, Zhang Y, Shen Y, Chen Y, Shi T, Yang H, Wang Z, Yan R
Sci Adv (2024) 10 pp. eadl3685-eadl3685 [ DOI: doi:10.1126/sciadv.adl3685 Pubmed: 38552027 ]
- 1,2-diacyl-glycerol-3-sn-phosphate (704 Da, Ligand)
- Water (18 Da, Ligand)
- Cholesterol hemisuccinate (486 Da, Ligand)
- Solute carrier family 13 member 2 (65 kDa, Protein from Homo sapiens)
- Sodium ion (22 Da, Ligand)
- Citric acid (192 Da, Ligand)
- Structure of nadc1 in complex with citrate (Complex from Homo sapiens)
CryoEM structure of NaDC1 in apo state
Resolution: 2.5 Å
EM Method: Single-particle
Fitted PDBs: 8w6d
Q-score: 0.662
Chi X, Chen Y, Li Y, Dai L, Zhang Y, Shen Y, Chen Y, Shi T, Yang H, Wang Z, Yan R
Sci Adv (2024) 10 pp. eadl3685-eadl3685 [ DOI: doi:10.1126/sciadv.adl3685 Pubmed: 38552027 ]
- 1,2-diacyl-glycerol-3-sn-phosphate (704 Da, Ligand)
- Cholesterol hemisuccinate (486 Da, Ligand)
- Structure of nadc1 in apo state (Complex from Homo sapiens)
- Solute carrier family 13 member 2 (65 kDa, Protein from Homo sapiens)
- Sodium ion (22 Da, Ligand)
Resolution: 3.3 Å
EM Method: Single-particle
Fitted PDBs: 8w6g
Q-score: 0.552
Chi X, Chen Y, Li Y, Dai L, Zhang Y, Shen Y, Chen Y, Shi T, Yang H, Wang Z, Yan R
Sci Adv (2024) 10 pp. eadl3685-eadl3685 [ DOI: doi:10.1126/sciadv.adl3685 Pubmed: 38552027 ]
- 2-[[(~{e})-3-(4-pentylphenyl)prop-2-enoyl]amino]benzoic acid (337 Da, Ligand)
- 1,2-diacyl-glycerol-3-sn-phosphate (704 Da, Ligand)
- Nadc1 in complex with inhibitor n-(p-amylcinnamoyl)anthranilic acid (aca) (Complex from Homo sapiens)
- Cholesterol hemisuccinate (486 Da, Ligand)
- Solute carrier family 13 member 2 (65 kDa, Protein from Homo sapiens)
NaS1 with sulfate - IN/IN state
Resolution: 3.1 Å
EM Method: Single-particle
Fitted PDBs: 8w6h
Q-score: 0.567
Chi X, Chen Y, Li Y, Dai L, Zhang Y, Shen Y, Chen Y, Shi T, Yang H, Wang Z, Yan R
Sci Adv (2024) 10 pp. eadl3685-eadl3685 [ DOI: doi:10.1126/sciadv.adl3685 Pubmed: 38552027 ]
- Sulfate ion (96 Da, Ligand)
- Solute carrier family 13 member 1 (67 kDa, Protein from Homo sapiens)
- Dimer of nas1 with sulfate in in/in state (Complex from Homo sapiens)
- Sodium ion (22 Da, Ligand)
- Cholesterol (386 Da, Ligand)
NaS1 with sulfate in IN/OUT state
Resolution: 3.2 Å
EM Method: Single-particle
Fitted PDBs: 8w6n
Q-score: 0.536
Chi X, Chen Y, Li Y, Dai L, Zhang Y, Shen Y, Chen Y, Shi T, Yang H, Wang Z, Yan R
Sci Adv (2024) 10 pp. eadl3685-eadl3685 [ DOI: doi:10.1126/sciadv.adl3685 Pubmed: 38552027 ]
- Sodium ion (22 Da, Ligand)
- Sulfate ion (96 Da, Ligand)
- Solute carrier family 13 member 1 (67 kDa, Protein from Homo sapiens)
- Structure of nas1 in complex with sulfate (Complex from Homo sapiens)
Resolution: 2.9 Å
EM Method: Single-particle
Fitted PDBs: 8w6o
Q-score: 0.58
Chi X, Chen Y, Li Y, Dai L, Zhang Y, Shen Y, Chen Y, Shi T, Yang H, Wang Z, Yan R
Sci Adv (2024) 10 pp. eadl3685-eadl3685 [ DOI: doi:10.1126/sciadv.adl3685 Pubmed: 38552027 ]
- Cholesterol (386 Da, Ligand)
- Sodium ion (22 Da, Ligand)
- Solute carrier family 13 member 1 (67 kDa, Protein from Homo sapiens)
- Dimer of nas1 in in/in state (Complex from Homo sapiens)
Resolution: 3.0 Å
EM Method: Single-particle
Fitted PDBs: 8w6t
Q-score: 0.54
Chi X, Chen Y, Li Y, Dai L, Zhang Y, Shen Y, Chen Y, Shi T, Yang H, Wang Z, Yan R
Sci Adv (2024) 10 pp. eadl3685-eadl3685 [ DOI: doi:10.1126/sciadv.adl3685 Pubmed: 38552027 ]
- Dimer of nas1 in in/out state (Complex from Homo sapiens)
- Solute carrier family 13 member 1 (67 kDa, Protein from Homo sapiens)
Structure of Calcium-Sensing Receptor in complex with NPS-2143
Resolution: 3.2 Å
EM Method: Single-particle
Fitted PDBs: 7dd5
Q-score: 0.415
Wen T, Wang Z, Chen X, Ren Y, Lu X, Xing Y, Lu J, Chang S, Zhang X, Shen Y, Yang X
Sci Adv (2021) 7 [ DOI: doi:10.1126/sciadv.abg1483 Pubmed: 34088669 ]
- Water (18 Da, Ligand)
- Tryptophan (204 Da, Ligand)
- Chloride ion (35 Da, Ligand)
- Calcium-sensing receptor (119 kDa, Protein from Gallus gallus)
- 2-chloro-6-[(2r)-2-hydroxy-3-{[2-methyl-1-(naphthalen-2-yl)propan-2-yl]amino}propoxy]benzonitrile (408 Da, Ligand)
- Calcium ion (40 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Calcium-sensing receptor from gallus gallus with ca2+/l-trp/nps-2143 (Cell from Gallus gallus)
Structure of Ca2+/L-Trp-bonnd Calcium-Sensing Receptor in active state
Resolution: 3.2 Å
EM Method: Single-particle
Fitted PDBs: 7dd6
Q-score: 0.41
Wen T, Wang Z, Chen X, Ren Y, Lu X, Xing Y, Lu J, Chang S, Zhang X, Shen Y, Yang X
Sci Adv (2021) 7 [ DOI: doi:10.1126/sciadv.abg1483 Pubmed: 34088669 ]
- Tryptophan (204 Da, Ligand)
- Chloride ion (35 Da, Ligand)
- Calcium-sensing receptor from gallus gallus with ca2+ and l-trp (Cell from Gallus gallus)
- Calcium-sensing receptor (119 kDa, Protein from Gallus gallus)
- Calcium ion (40 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Structure of Calcium-Sensing Receptor in complex with Evocalcet
Resolution: 3.2 Å
EM Method: Single-particle
Fitted PDBs: 7dd7
Q-score: 0.414
Wen T, Wang Z, Chen X, Ren Y, Lu X, Xing Y, Lu J, Chang S, Zhang X, Shen Y, Yang X
Sci Adv (2021) 7 [ DOI: doi:10.1126/sciadv.abg1483 Pubmed: 34088669 ]
- Calcium-sensing receptor in complex with evocalcet (Cell from Gallus gallus)
- Tryptophan (204 Da, Ligand)
- Chloride ion (35 Da, Ligand)
- 2-[4-[(3s)-3-[[(1r)-1-naphthalen-1-ylethyl]amino]pyrrolidin-1-yl]phenyl]ethanoic acid (374 Da, Ligand)
- Calcium-sensing receptor (119 kDa, Protein from Gallus gallus)
- Calcium ion (40 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)