Lysophosphatidic acid receptor 1-Gi complex bound to LPA
Resolution: 2.83 Å
EM Method: Single-particle
Fitted PDBs: 7td0
Q-score: 0.527
Liu S, Paknejad N, Zhu L, Kihara Y, Ray M, Chun J, Liu W, Hite RK, Huang XY
Nat Commun (2022) 13 pp. 731-731 [ Pubmed: 35136060 DOI: doi:10.1038/s41467-022-28417-2 ]
- Lysophosphatidic acid receptor 1 (39 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Bos taurus)
- Guanine nucleotide-binding protein g(i) subunit alpha-1 (43 kDa, Protein from Rattus norvegicus)
- Complex of lysophosphatidic acid receptor 1 with g-protein and lpa (Complex from Bos taurus)
- (2r)-2-hydroxy-3-(phosphonooxy)propyl (9e)-octadec-9-enoate (436 Da, Ligand)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (37 kDa, Protein from Bos taurus)
Lysophosphatidic acid receptor 1-Gi complex bound to LPA, state a
Resolution: 3.08 Å
EM Method: Single-particle
Fitted PDBs: 7td1
Q-score: 0.496
Liu S, Paknejad N, Zhu L, Kihara Y, Ray M, Chun J, Liu W, Hite RK, Huang XY
Nat Commun (2022) 13 pp. 731-731 [ Pubmed: 35136060 DOI: doi:10.1038/s41467-022-28417-2 ]
- Lysophosphatidic acid receptor 1 (39 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Bos taurus)
- Guanine nucleotide-binding protein g(i) subunit alpha-1 (43 kDa, Protein from Rattus norvegicus)
- Complex of lysophosphatidic acid receptor 1 with g-protein and lpa (Complex from Bos taurus)
- (2r)-2-hydroxy-3-(phosphonooxy)propyl (9e)-octadec-9-enoate (436 Da, Ligand)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (37 kDa, Protein from Bos taurus)
Lysophosphatidic acid receptor 1-Gi complex bound to LPA, state a
Resolution: 3.11 Å
EM Method: Single-particle
Fitted PDBs: 7td2
Q-score: 0.506
Liu S, Paknejad N, Zhu L, Kihara Y, Ray M, Chun J, Liu W, Hite RK, Huang XY
Nat Commun (2022) 13 pp. 731-731 [ Pubmed: 35136060 DOI: doi:10.1038/s41467-022-28417-2 ]
- Lysophosphatidic acid receptor 1 (39 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Bos taurus)
- Guanine nucleotide-binding protein g(i) subunit alpha-1 (43 kDa, Protein from Rattus norvegicus)
- Complex of lysophosphatidic acid receptor 1 with g-protein and lpa (Complex from Bos taurus)
- (2r)-2-hydroxy-3-(phosphonooxy)propyl (9e)-octadec-9-enoate (436 Da, Ligand)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (37 kDa, Protein from Bos taurus)
Sphingosine-1-phosphate receptor 1-Gi complex bound to S1P
Resolution: 3.0 Å
EM Method: Single-particle
Fitted PDBs: 7td3
Q-score: 0.574
Liu S, Paknejad N, Zhu L, Kihara Y, Ray M, Chun J, Liu W, Hite RK, Huang XY
Nat Commun (2022) 13 pp. 731-731 [ Pubmed: 35136060 DOI: doi:10.1038/s41467-022-28417-2 ]
- (2s,3r,4e)-2-amino-3-hydroxyoctadec-4-en-1-yl dihydrogen phosphate (379 Da, Ligand)
- Complex of sphingosine-1-phosphate receptor 1 with g-protein and s1p (Complex from Bos taurus)
- Sphingosine 1-phosphate receptor 1 (43 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Bos taurus)
- Guanine nucleotide-binding protein g(i) subunit alpha-1 (43 kDa, Protein from Rattus norvegicus)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (37 kDa, Protein from Bos taurus)
Sphingosine-1-phosphate receptor 1-Gi complex bound to Siponimod
Resolution: 2.6 Å
EM Method: Single-particle
Fitted PDBs: 7td4
Q-score: 0.605
Liu S, Paknejad N, Zhu L, Kihara Y, Ray M, Chun J, Liu W, Hite RK, Huang XY
Nat Commun (2022) 13 pp. 731-731 [ Pubmed: 35136060 DOI: doi:10.1038/s41467-022-28417-2 ]
- Sphingosine 1-phosphate receptor 1 (43 kDa, Protein from Homo sapiens)
- Complex of sphingosine-1-phosphate receptor 1 with g-protein and siponimod (Complex from Bos taurus)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Bos taurus)
- Guanine nucleotide-binding protein g(i) subunit alpha-1 (43 kDa, Protein from Rattus norvegicus)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- 1-[[4-[(~{e})-~{n}-[[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy]-~{c}-methyl-carbonimidoyl]-2-ethyl-phenyl]methyl]azetidine-3-carboxylic acid (516 Da, Ligand)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (37 kDa, Protein from Bos taurus)