Resolution: 3.5 Å
EM Method: Single-particle
Fitted PDBs: 8t6j
Q-score: 0.463
Krishna Kumar K, Wang H, Habrian C, Latorraca NR, Xu J, O'Brien ES, Zhang C, Montabana E, Koehl A, Marqusee S, Isacoff EY, Kobilka BK
Nature (2024) 629 pp. 951-956 [ DOI: doi:10.1038/s41586-024-07327-x Pubmed: 38632403 ]
Resolution: 3.3 Å
EM Method: Single-particle
Fitted PDBs: 8t7h
Q-score: 0.43
Krishna Kumar K, Wang H, Habrian C, Latorraca NR, Xu J, O'Brien ES, Zhang C, Montabana E, Koehl A, Marqusee S, Isacoff EY, Kobilka BK
Nature (2024) 629 pp. 951-956 [ DOI: doi:10.1038/s41586-024-07327-x Pubmed: 38632403 ]
- Metabotropic glutamate receptor 5 in complex with quis (Cellular component from Homo sapiens)
- Nanobody 43 (13 kDa, Protein from Lama glama)
- (s)-2-amino-3-(3,5-dioxo-[1,2,4]oxadiazolidin-2-yl)-propionic acid (189 Da, Ligand)
- Metabotropic glutamate receptor 5 (98 kDa, Protein from Homo sapiens)
Resolution: 3.0 Å
EM Method: Single-particle
Fitted PDBs: 8t8m
Q-score: 0.493
Krishna Kumar K, Wang H, Habrian C, Latorraca NR, Xu J, O'Brien ES, Zhang C, Montabana E, Koehl A, Marqusee S, Isacoff EY, Kobilka BK
Nature (2024) 629 pp. 951-956 [ DOI: doi:10.1038/s41586-024-07327-x Pubmed: 38632403 ]
- Metabotropic glutamate receptor 5 in complex with quis (Cellular component from Homo sapiens)
- (s)-2-amino-3-(3,5-dioxo-[1,2,4]oxadiazolidin-2-yl)-propionic acid (189 Da, Ligand)
- Metabotropic glutamate receptor 5 (98 kDa, Protein from Homo sapiens)
- Nb43 (13 kDa, Protein from Lama glama)
Quis and CDPPB bound active mGlu5
Resolution: 2.9 Å
EM Method: Single-particle
Fitted PDBs: 8tao
Q-score: 0.486
Krishna Kumar K, Wang H, Habrian C, Latorraca NR, Xu J, O'Brien ES, Zhang C, Montabana E, Koehl A, Marqusee S, Isacoff EY, Kobilka BK
Nature (2024) 629 pp. 951-956 [ DOI: doi:10.1038/s41586-024-07327-x Pubmed: 38632403 ]
- 3-cyano-n-(1,3-diphenyl-1h-pyrazol-5-yl)benzamide (364 Da, Ligand)
- Metabotropic glutamate receptor 5 (98 kDa, Protein from Homo sapiens)
- Nb43 (13 kDa, Protein from Lama glama)
- Metabotropic glutamate receptor 5 bound to quis and cdppb, in complex with nb43 (Cellular component from Homo sapiens)
- (s)-2-amino-3-(3,5-dioxo-[1,2,4]oxadiazolidin-2-yl)-propionic acid (189 Da, Ligand)
GCGR-Gs complex in the presence of RAMP2
Resolution: 2.9 Å
EM Method: Single-particle
Fitted PDBs: 8fu6
Q-score: 0.543
Krishna Kumar K, O'Brien ES, Habrian CH, Latorraca NR, Wang H, Tuneew I, Montabana E, Marqusee S, Hilger D, Isacoff EY, Mathiesen JM, Kobilka BK
Cell (2023) 186 pp. 1465-1477.e18 [ Pubmed: 37001505 DOI: doi:10.1016/j.cell.2023.02.028 ]
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (39 kDa, Protein from Homo sapiens)
- Nb35 (15 kDa, Protein from Lama glama)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Homo sapiens)
- Gcgr-gs signaling complex in the presence of ramp2 (Complex from Homo sapiens)
- Guanine nucleotide-binding protein g(s) subunit alpha isoforms short (44 kDa, Protein from Homo sapiens)
- Glucagon derivative zp3780 (3 kDa, Protein from synthetic construct)
- Glucagon receptor (56 kDa, Protein from Homo sapiens)