Resolution: 2.75 Å
EM Method: Single-particle
Fitted PDBs: 8wgr
Q-score: 0.576
Tan J, Xiao Y, Kong F, Zhang X, Xu H, Zhu A, Liu Y, Lei J, Tian B, Yuan Y, Yan C
Nature (2024) 632 pp. 921-929 [ DOI: doi:10.1038/s41586-024-07719-z Pubmed: 39048818 ]
- Water (18 Da, Ligand)
- Potassium ion (39 Da, Ligand)
- Net (110 kDa, Complex from Homo sapiens)
- Sodium-dependent noradrenaline transporter (69 kDa, Protein from Homo sapiens)
- Chloride ion (35 Da, Ligand)
- 3-(10,11-dihydro-5h-dibenzo[b,f]azepin-5-yl)-n-methylpropan-1-amine (266 Da, Ligand)
Resolution: 3.47 Å
EM Method: Single-particle
Fitted PDBs: 8wgx
Q-score: 0.462
Tan J, Xiao Y, Kong F, Zhang X, Xu H, Zhu A, Liu Y, Lei J, Tian B, Yuan Y, Yan C
Nature (2024) 632 pp. 921-929 [ DOI: doi:10.1038/s41586-024-07719-z Pubmed: 39048818 ]
- Sodium-dependent noradrenaline transporter (69 kDa, Protein from Homo sapiens)
- L-norepinephrine (169 Da, Ligand)
- Net (110 kDa, Complex from Homo sapiens)
Resolution: 3.4 Å
EM Method: Single-particle
Fitted PDBs: 8z1l
Q-score: 0.451
Tan J, Xiao Y, Kong F, Zhang X, Xu H, Zhu A, Liu Y, Lei J, Tian B, Yuan Y, Yan C
Nature (2024) 632 pp. 921-929 [ DOI: doi:10.1038/s41586-024-07719-z Pubmed: 39048818 ]
- Sodium-dependent noradrenaline transporter (69 kDa, Protein from Homo sapiens)
- (3r)-n-methyl-3-(2-methylphenoxy)-3-phenyl-propan-1-amine (255 Da, Ligand)
- Chloride ion (35 Da, Ligand)
- Net (110 kDa, Complex from Homo sapiens)
Resolution: 2.85 Å
EM Method: Single-particle
Fitted PDBs: 8i3v
Q-score: 0.57
Tan J, Xiao Y, Kong F, Zhang X, Xu H, Zhu A, Liu Y, Lei J, Tian B, Yuan Y, Yan C
Nature (2024) 632 pp. 921-929 [ DOI: doi:10.1038/s41586-024-07719-z Pubmed: 39048818 ]
- Water (18 Da, Ligand)
- (1s)-1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3-dihydro-2-benzofuran-5-carbonitrile (324 Da, Ligand)
- Sodium-dependent noradrenaline transporter (69 kDa, Protein from Homo sapiens)
- Chloride ion (35 Da, Ligand)
- Net (Complex from Homo sapiens)
Resolution: 2.5 Å
EM Method: Single-particle
Fitted PDBs: 8hfe
Q-score: 0.629
Tan J, Xiao Y, Kong F, Zhang X, Xu H, Zhu A, Liu Y, Lei J, Tian B, Yuan Y, Yan C
Nature (2024) 632 pp. 921-929 [ DOI: doi:10.1038/s41586-024-07719-z Pubmed: 39048818 ]
- Sodium-dependent noradrenaline transporter (69 kDa, Protein from Homo sapiens)
- Water (18 Da, Ligand)
- Chloride ion (35 Da, Ligand)
- Net (110 kDa, Complex from Homo sapiens)
Resolution: 2.86 Å
EM Method: Single-particle
Fitted PDBs: 8hff
Q-score: 0.537
Tan J, Xiao Y, Kong F, Zhang X, Xu H, Zhu A, Liu Y, Lei J, Tian B, Yuan Y, Yan C
Nature (2024) 632 pp. 921-929 [ DOI: doi:10.1038/s41586-024-07719-z Pubmed: 39048818 ]
- Sodium-dependent noradrenaline transporter (69 kDa, Protein from Homo sapiens)
- L-norepinephrine (169 Da, Ligand)
- Water (18 Da, Ligand)
- Net (110 kDa, Complex from Homo sapiens)
Resolution: 3.0 Å
EM Method: Single-particle
Fitted PDBs: 8hfg
Q-score: 0.442
Tan J, Xiao Y, Kong F, Zhang X, Xu H, Zhu A, Liu Y, Lei J, Tian B, Yuan Y, Yan C
Nature (2024) 632 pp. 921-929 [ DOI: doi:10.1038/s41586-024-07719-z Pubmed: 39048818 ]
- Water (18 Da, Ligand)
- Net (110 kDa, Complex from Homo sapiens)
- Sodium-dependent noradrenaline transporter (69 kDa, Protein from Homo sapiens)
- Chloride ion (35 Da, Ligand)
- L-dopamine (153 Da, Ligand)
Resolution: 2.5 Å
EM Method: Single-particle
Fitted PDBs: 8hfi
Q-score: 0.644
Tan J, Xiao Y, Kong F, Zhang X, Xu H, Zhu A, Liu Y, Lei J, Tian B, Yuan Y, Yan C
Nature (2024) 632 pp. 921-929 [ DOI: doi:10.1038/s41586-024-07719-z Pubmed: 39048818 ]
- Water (18 Da, Ligand)
- Net (110 kDa, Complex from Homo sapiens)
- Sodium-dependent noradrenaline transporter (69 kDa, Protein from Homo sapiens)
- Chloride ion (35 Da, Ligand)
- 3-(10,11-dihydro-5h-dibenzo[b,f]azepin-5-yl)-n-methylpropan-1-amine (266 Da, Ligand)
Resolution: 3.0 Å
EM Method: Single-particle
Fitted PDBs: 8hfl
Q-score: 0.556
Tan J, Xiao Y, Kong F, Zhang X, Xu H, Zhu A, Liu Y, Lei J, Tian B, Yuan Y, Yan C
Nature (2024) 632 pp. 921-929 [ DOI: doi:10.1038/s41586-024-07719-z Pubmed: 39048818 ]
- Water (18 Da, Ligand)
- Bupropion (239 Da, Ligand)
- Net (110 kDa, Complex from Homo sapiens)
- Sodium-dependent noradrenaline transporter (69 kDa, Protein from Homo sapiens)
- Chloride ion (35 Da, Ligand)
Cryo-EM structure of human apo GABA transporter GAT1 in an inward-open state
Resolution: 2.2 Å
EM Method: Single-particle
Fitted PDBs: 7y7v
Q-score: 0.681
Zhu A, Huang J, Kong F, Tan J, Lei J, Yuan Y, Yan C
Nat Struct Mol Biol (2023) 30 pp. 1012-1022 [ DOI: doi:10.1038/s41594-023-00983-z Pubmed: 37400655 ]
- Water (18 Da, Ligand)
- Gat1 (110 kDa, Complex from Homo sapiens)
- Sodium- and chloride-dependent gaba transporter 1 (70 kDa, Protein from Homo sapiens)
- Chloride ion (35 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)