Cryo-EM structure of ACE2-SIT1 complex with tiagabine
Resolution: 3.34 Å
EM Method: Single-particle
Fitted PDBs: 8wm3
Q-score: 0.366
Broer A, Hu Z, Kukulowicz J, Yadav A, Zhang T, Dai L, Bajda M, Yan R, Broer S
J Biol Chem (2024) 300 pp. 107687-107687 [ DOI: doi:10.1016/j.jbc.2024.107687 Pubmed: 39159813 ]
- Sodium- and chloride-dependent transporter xtrp3 (68 kDa, Protein from Homo sapiens)
- Tiagabine (375 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Angiotensin-converting enzyme 2 (94 kDa, Protein from Homo sapiens)
- Ace2-sit1 compelx with tiagabine (Complex from Homo sapiens)
Cryo-EM structure of ACE2-B0AT1 complex with JX98
Xu J, Hu Z, Dai L, Yadav A, Jiang Y, Broer A, Gardiner MG, McLeod M, Yan R, Broer S
Nat Commun (2024) 15 pp. 7224-7224 [ DOI: doi:10.1038/s41467-024-51748-1 Pubmed: 39174516 ]
- Ace2-b0at1 complex with inhibitor jx98 (Complex from Homo sapiens)
- 2-(4-chloranyl-3,5-dimethyl-phenoxy)-~{n}-propan-2-yl-ethanamide (255 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Sodium-dependent neutral amino acid transporter b(0)at1 (72 kDa, Protein from Homo sapiens)
- Angiotensin-converting enzyme 2 (94 kDa, Protein from Homo sapiens)
Cryo-EM structure of ACE2-B0AT1 complex with JX225
Resolution: 3.2 Å
EM Method: Single-particle
Fitted PDBs: 8wbz
Q-score: 0.466
Xu J, Hu Z, Dai L, Yadav A, Jiang Y, Broer A, Gardiner MG, McLeod M, Yan R, Broer S
Nat Commun (2024) 15 pp. 7224-7224 [ DOI: doi:10.1038/s41467-024-51748-1 Pubmed: 39174516 ]
- Ace2-b0at1 complex with inhibitor jx225 (Complex from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Sodium-dependent neutral amino acid transporter b(0)at1 (72 kDa, Protein from Homo sapiens)
- 2-(4-bromanyl-3-methyl-phenoxy)-~{n}-propyl-ethanamide (286 Da, Ligand)
- Angiotensin-converting enzyme 2 (94 kDa, Protein from Homo sapiens)
Cryo EM map of SLC7A10 in the apo state
Resolution: 3.42 Å
EM Method: Single-particle
Fitted PDBs: 8wns
Q-score: 0.406
Li Y, Guo Y, Broer A, Dai L, Broer S, Yan R
Nat Commun (2024) 15 pp. 3036-3036 [ Pubmed: 38589439 DOI: doi:10.1038/s41467-024-47468-1 ]
- Amino acid transporter heavy chain slc3a2 (68 kDa, Protein from Homo sapiens)
- Asc-type amino acid transporter 1 (56 kDa, Protein from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- 4f2hc-asc-1 complex (Complex from Homo sapiens)
Cryo EM map of SLC7A10 with L-Alanine substrate
Resolution: 3.42 Å
EM Method: Single-particle
Fitted PDBs: 8wnt
Q-score: 0.425
Li Y, Guo Y, Broer A, Dai L, Yan R
Nat Commun (2024) 15 pp. 3036-3036 [ Pubmed: 38589439 DOI: doi:10.1038/s41467-024-47468-1 ]
- Asc-type amino acid transporter 1 (56 kDa, Protein from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- 4f2hc-asc-1 complex (Complex from Homo sapiens)
- Amino acid transporter heavy chain slc3a2 (68 kDa, Protein from Homo sapiens)
- Alanine (89 Da, Ligand)
Cryo EM map of SLC7A10-SLC3A2 complex in the D-serine bound state
Resolution: 3.5 Å
EM Method: Single-particle
Fitted PDBs: 8wny
Q-score: 0.456
Li Y, Guo Y, Broer A, Dai L, Yan R
Nat Commun (2024) 15 pp. 3036-3036 [ Pubmed: 38589439 DOI: doi:10.1038/s41467-024-47468-1 ]
- Asc-type amino acid transporter 1 (56 kDa, Protein from Homo sapiens)
- D-serine (105 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- 4f2hc-asc-1 complex (Complex from Homo sapiens)
- Amino acid transporter heavy chain slc3a2 (68 kDa, Protein from Homo sapiens)