Syrjanen JL, Michalski K, Chou TH, Grant T, Rao S, Simorowski N, Tucker SJ, Grigorieff N, Furukawa H
Nat. Struct. Mol. Biol. (2020) 27 pp. 150-159 [ Pubmed: 31988524 DOI: 10.1038/s41594-019-0369-9 ]
Image sets:
Chicken CALHM1 - Human CALHM2 chimera
Syrjanen JL, Michalski K, Chou TH, Grant T, Rao S, Simorowski N, Tucker SJ, Grigorieff N, Furukawa H
Nat. Struct. Mol. Biol. (2020) 27 pp. 150-159 [ Pubmed: 31988524 DOI: 10.1038/s41594-019-0369-9 ]
Image sets:
Human CALHM2 gap junction in nanodisc, 1 mM CaCl2 and 1 mM ATP
Syrjanen JL, Michalski K, Chou TH, Grant T, Rao S, Simorowski N, Tucker SJ, Grigorieff N, Furukawa H
Nat. Struct. Mol. Biol. (2020) 27 pp. 150-159 [ Pubmed: 31988524 DOI: 10.1038/s41594-019-0369-9 ]
Image sets:
Human CALHM2 in nanodisc, 1 mM EDTA
Syrjanen JL, Michalski K, Chou TH, Grant T, Rao S, Simorowski N, Tucker SJ, Grigorieff N, Furukawa H
Nat. Struct. Mol. Biol. (2020) 27 pp. 150-159 [ Pubmed: 31988524 DOI: 10.1038/s41594-019-0369-9 ]
Image sets:
GluN1b-GluN2B NMDA receptor in non-active 2 conformation at 4 angstrom resolution
Resolution: 3.99 Å
EM Method: Single-particle
Fitted PDBs: 6whr
Q-score: 0.411
Chou TH, Tajima N, Romero-Hernandez A, Furukawa H
Cell (2020) 182 pp. 357-371.e13 [ Pubmed: 32610085 DOI: doi:10.1016/j.cell.2020.05.052 ]
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Rattus norvegicus)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Nmda receptor glun1b/2b functional ion channel complex (Complex from Rattus norvegicus)
- Glutamate receptor ionotropic, nmda 1 (108 kDa, Protein from Rattus norvegicus)
GluN1b-GluN2B NMDA receptor in non-active 1 conformation at 3.95 angstrom resolution
Resolution: 4.0 Å
EM Method: Single-particle
Fitted PDBs: 6whs
Q-score: 0.421
Chou TH, Tajima N, Romero-Hernandez A, Furukawa H
Cell (2020) 182 pp. 357-371.e13 [ DOI: doi:10.1016/j.cell.2020.05.052 Pubmed: 32610085 ]
- Glutamate receptor ionotropic, nmda 1 (108 kDa, Protein from Rattus norvegicus)
- Nmda receptor glun1b/2b functional ion channel complex (Complex from Rattus norvegicus)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Rattus norvegicus)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
GluN1b-GluN2B NMDA receptor in active conformation at 4.4 angstrom resolution
Resolution: 4.39 Å
EM Method: Single-particle
Fitted PDBs: 6wht
Q-score: 0.35
Chou TH, Tajima N, Romero-Hernandez A, Furukawa H
Cell (2020) 182 pp. 357-371.e13 [ DOI: doi:10.1016/j.cell.2020.05.052 Pubmed: 32610085 ]
- Glutamate receptor ionotropic, nmda 1 (108 kDa, Protein from Rattus norvegicus)
- Nmda receptor glun1b/2b functional ion channel complex (Complex from Rattus norvegicus)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Rattus norvegicus)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
GluN1b-GluN2B NMDA receptor in complex with SDZ 220-040 and L689,560, class 1
Resolution: 3.93 Å
EM Method: Single-particle
Fitted PDBs: 6whu
Q-score: 0.42
Chou TH, Tajima N, Romero-Hernandez A, Furukawa H
Cell (2020) 182 pp. 357-371.e13 [ DOI: doi:10.1016/j.cell.2020.05.052 Pubmed: 32610085 ]
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Rattus norvegicus)
- (2s)-2-amino-3-[2',4'-dichloro-4-hydroxy-5-(phosphonomethyl)biphenyl-3-yl]propanoic acid (420 Da, Ligand)
- Nmda receptor glun1b/2b functional ion channel complex (Complex from Rattus norvegicus)
- (2r,4s)-5,7-dichloro-4-[(phenylcarbamoyl)amino]-1,2,3,4-tetrahydroquinoline-2-carboxylic acid (380 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Glutamate receptor ionotropic, nmda 1 (108 kDa, Protein from Rattus norvegicus)
GluN1b-GluN2B NMDA receptor in complex with SDZ 220-040 and L689,560, class 2
Resolution: 4.05 Å
EM Method: Single-particle
Fitted PDBs: 6whv
Q-score: 0.394
Chou TH, Tajima N, Romero-Hernandez A, Furukawa H
Cell (2020) 182 pp. 357-371.e13 [ DOI: doi:10.1016/j.cell.2020.05.052 Pubmed: 32610085 ]
- (2s)-2-amino-3-[2',4'-dichloro-4-hydroxy-5-(phosphonomethyl)biphenyl-3-yl]propanoic acid (420 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Rattus norvegicus)
- Nmda receptor glun1b/2b functional ion channel complex (Complex from Rattus norvegicus)
- (2r,4s)-5,7-dichloro-4-[(phenylcarbamoyl)amino]-1,2,3,4-tetrahydroquinoline-2-carboxylic acid (380 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Glutamate receptor ionotropic, nmda 1 (108 kDa, Protein from Rattus norvegicus)
GluN1b-GluN2B NMDA receptor in complex with GluN2B antagonist SDZ 220-040, class 1
Resolution: 4.09 Å
EM Method: Single-particle
Fitted PDBs: 6whw
Q-score: 0.454
Chou TH, Tajima N, Romero-Hernandez A, Furukawa H
Cell (2020) 182 pp. 357-371.e13 [ DOI: doi:10.1016/j.cell.2020.05.052 Pubmed: 32610085 ]
- (2s)-2-amino-3-[2',4'-dichloro-4-hydroxy-5-(phosphonomethyl)biphenyl-3-yl]propanoic acid (420 Da, Ligand)
- Nmda receptor glun1b/2b functional ion channel complex (Complex from Rattus norvegicus)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Ionotropic glutamate receptor , nmda receptor glun1b (108 kDa, Protein from Rattus norvegicus)
- Ionotropic glutamate receptor , nmda receptor glun2b (98 kDa, Protein from Rattus norvegicus)