Resolution: 2.91 Å
EM Method: Single-particle
Fitted PDBs: 9jmz
Q-score: 0.489
Song H, Hao T, Han P, Wang H, Zhang X, Li X, Wang Y, Chen J, Li Y, Jin X, Duan X, Zhang W, Bi Y, Jin R, Sun L, Wang N, Gao GF
Cell (2025) [ Pubmed: 39848246 DOI: doi:10.1016/j.cell.2025.01.019 ]
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Human-infecting bovine influenza h5n1 hemagglutinin complexed with avian receptor analog lsta (Complex from Influenza A virus (A/Indonesia/5/2005(H5N1)))
- N-acetyl-alpha-neuraminic acid (309 Da, Ligand)
- Hemagglutinin (57 kDa, Protein from Influenza A virus (A/Indonesia/5/2005(H5N1)))
Structure of wild type human PSS1
Long T, Li D, Vale G, Jiang Y, Schmiege P, Yang ZJ, McDonald JG, Li X
Cell (2024) 187 pp. 5665-5678.e18 [ Pubmed: 39208797 DOI: doi:10.1016/j.cell.2024.08.004 ]
- Water (18 Da, Ligand)
- Pss1 (Complex from Homo sapiens)
- (2r)-3-{[(s)-hydroxy{[(1r,2r,3r,4r,5r,6s)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propane-1,2-diyl dihexadecanoate (811 Da, Ligand)
- 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine (760 Da, Ligand)
- Calcium ion (40 Da, Ligand)
- O-[(r)-{[(2r)-2,3-bis(octadecanoyloxy)propyl]oxy}(hydroxy)phosphoryl]-l-serine (792 Da, Ligand)
- [(2~{r})-1-[2-azanylethoxy(oxidanyl)phosphoryl]oxy-3-hexadecanoyloxy-propan-2-yl] (~{z})-octadec-9-enoate (717 Da, Ligand)
- Phosphatidylserine synthase 1 (48 kDa, Protein from Homo sapiens)
Long T, Li D, Vale G, Jiang Y, Schmiege P, Yang ZJ, McDonald JG, Li X
Cell (2024) 187 pp. 5665-5678.e18 [ Pubmed: 39208797 DOI: doi:10.1016/j.cell.2024.08.004 ]
- Phosphatidylserine synthase 1 (56 kDa, Protein from Homo sapiens)
- Calcium ion (40 Da, Ligand)
- Human pss1-p269s (Complex from Homo sapiens)
Structure of inhibitor-bound human PSS1
Long T, Li D, Vale G, Jiang Y, Schmiege P, Yang ZJ, McDonald JG, Li X
Cell (2024) 187 pp. 5665-5678.e18 [ Pubmed: 39208797 DOI: doi:10.1016/j.cell.2024.08.004 ]
- Water (18 Da, Ligand)
- (2r)-3-{[(s)-hydroxy{[(1r,2r,3r,4r,5r,6s)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propane-1,2-diyl dihexadecanoate (811 Da, Ligand)
- 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine (760 Da, Ligand)
- Calcium ion (40 Da, Ligand)
- Inhibitor-bound human pss1 (Complex from Homo sapiens)
- (7p)-7-[(4s)-4-{4-[3,5-bis(trifluoromethyl)phenoxy]phenyl}-5-(2,2-difluoropropyl)-6-oxo-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl]-1,3-benzoxazol-2(3h)-one (638 Da, Ligand)
- O-[(r)-{[(2r)-2,3-bis(octadecanoyloxy)propyl]oxy}(hydroxy)phosphoryl]-l-serine (792 Da, Ligand)
- [(2~{r})-1-[2-azanylethoxy(oxidanyl)phosphoryl]oxy-3-hexadecanoyloxy-propan-2-yl] (~{z})-octadec-9-enoate (717 Da, Ligand)
- Phosphatidylserine synthase 1 (48 kDa, Protein from Homo sapiens)
human connexin-36 gap junction channel in complex with mefloquine
Resolution: 2.13 Å
EM Method: Single-particle
Fitted PDBs: 8qoj
Q-score: 0.657
Ding X, Aureli S, Vaithia A, Lavriha P, Schuster D, Khanppnavar B, Li X, Blum TB, Picotti P, Gervasio FL, Korkhov VM
Cell Discov (2024) 10 pp. 68-68 [ Pubmed: 38890333 DOI: doi:10.1038/s41421-024-00691-y ]
- Human connexin-36 gap junction channel in complex with mefloquine (Complex from Homo sapiens)
- Water (18 Da, Ligand)
- Gap junction delta-2 protein (37 kDa, Protein from Homo sapiens)
- (11r,12s)- mefloquine (378 Da, Ligand)
human connexin-36 gap junction channel
Resolution: 2.53 Å
EM Method: Single-particle
Fitted PDBs: 8r7p
Q-score: 0.62
Ding X, Aureli S, Vaithia A, Lavriha P, Schuster D, Khanppnavar B, Li X, Blum TB, Picotti P, Gervasio FL, Korkhov VM
Cell Discov (2024) 10 pp. 68-68 [ Pubmed: 38890333 DOI: doi:10.1038/s41421-024-00691-y ]
- Human connexin-36 gap junction channel (Complex from Homo sapiens)
- Water (18 Da, Ligand)
- Gap junction delta-2 protein (37 kDa, Protein from Homo sapiens)
human connexin-36 gap junction channel in complex with quinine
Resolution: 2.78 Å
EM Method: Single-particle
Fitted PDBs: 8r7q
Q-score: 0.602
Ding X, Aureli S, Vaithia A, Lavriha P, Schuster D, Khanppnavar B, Li X, Blum TB, Picotti P, Gervasio FL, Korkhov VM
Cell Discov (2024) 10 pp. 68-68 [ Pubmed: 38890333 DOI: doi:10.1038/s41421-024-00691-y ]
- Quinine (324 Da, Ligand)
- Gap junction delta-2 protein (37 kDa, Protein from Homo sapiens)
- Human connexin-36 gap junction channel in complex with quinine (Complex from Homo sapiens)
Cryo-EM structure of apo-GPR30-Gq complex structure
Resolution: 2.9 Å
EM Method: Single-particle
Fitted PDBs: 8xog
Q-score: 0.462
Liu H, Guo S, Dai A, Xu P, Li X, Huang S, He X, Wu K, Zhang X, Yang D, Xie X, Xu HE
Cell Res (2024) 34 pp. 530-533 [ Pubmed: 38744981 DOI: doi:10.1038/s41422-024-00963-y ]
- Water (18 Da, Ligand)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Homo sapiens)
- Gpr30-gq (Complex from Homo sapiens)
- G-protein coupled estrogen receptor 1 (42 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (38 kDa, Protein from Homo sapiens)
- Scfv16 (Complex from synthetic construct)
- Guanine nucleotide-binding protein g(q) subunit alpha-q (41 kDa, Protein from Homo sapiens)
- Gpr30-gq complex (Complex)
- Scfv16 (26 kDa, Protein from synthetic construct)
Cryo-EM structure of thehydroxycarboxylic acid receptor 2-Gi protein complex bound niacin
Resolution: 3.05 Å
EM Method: Single-particle
Fitted PDBs: 8j6l
Q-score: 0.4
Zhu S, Yuan Q, Li X, He X, Shen S, Wang D, Li J, Cheng X, Duan X, Xu HE, Duan J
Cell Rep (2023) 42 pp. 113406-113406 [ Pubmed: 37952153 DOI: doi:10.1016/j.celrep.2023.113406 ]
- Guanine nucleotide-binding protein g(i) subunit alpha-1 (40 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (40 kDa, Protein from Homo sapiens)
- Nicotinic acid (123 Da, Ligand)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Homo sapiens)
- Hydroxycarboxylic acid receptor 2,hydroxycarboxylic acid receptor 2 (56 kDa, Protein from Homo sapiens)
- Complex of hydroxycarboxylic acid receptor 2 with mk-6892 (Complex from Homo sapiens)
- Svf16 (26 kDa, Protein from Homo sapiens)
PGF2-alpha bound Prostaglandin F2-alpha receptor-Gq Protein Complex
Resolution: 2.77 Å
EM Method: Single-particle
Fitted PDBs: 8xjl
Q-score: 0.559
Li X, Zhang X, Wen X, Zhang D, Qu C, Miao X, Zhang W, Zhang R, Liu G, Xiao P, Sun JP, Gong W
Cell Rep (2024) 43 pp. 113893-113893 [ Pubmed: 38446662 DOI: doi:10.1016/j.celrep.2024.113893 ]
- Pgf2-alpha-fp-minigq-scfv16 complex (Complex from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (40 kDa, Protein from Homo sapiens)
- Engineered minigq (28 kDa, Protein from synthetic construct)
- Antibody fragment scfv16 (27 kDa, Protein from synthetic construct)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Homo sapiens)
- (z)-7-[(1r,2r,3r,5s)-3,5-bis(oxidanyl)-2-[(e,3s)-3-oxidanyloct-1-enyl]cyclopentyl]hept-5-enoic acid (354 Da, Ligand)
- Fusion tag,prostaglandin f2-alpha receptor,lgbit (64 kDa, Protein from synthetic construct)