Zosuquidar and UIC2 Fab complex of human-mouse chimeric ABCB1 (ABCB1HM)
Resolution: 3.58 Å
EM Method: Single-particle
Fitted PDBs: 6fn1
Q-score: 0.442
Alam A, Kung R, Kowal J, McLeod RA, Tremp N, Broude EV, Roninson IB, Stahlberg H, Locher KP
PNAS (2018) 115 pp. E1973-E1982 [ DOI: doi:10.1073/pnas.1717044115 Pubmed: 29440498 ]
- Zosuquidar (527 Da, Ligand)
- Human-mouse chimeric abcb1 (abcbhm) (137 kDa, Protein from Homo sapiens)
- Human-mouse chimeric abcb1 (abcb1hm) complex with uic2 fab and zosuquidar (195 kDa, Complex)
- Human-mouse chimeric abcb1 (abcb1hm) complex with uic2 fab and zosuquidar (Complex from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Uic2 antigen binding fragment light chain (24 kDa, Protein from Mus musculus)
- Human-mouse chimeric abcb1 (abcb1hm) complex with uic2 fab and zosuquidar (Complex from Mus musculus)
- Uic2 antigen binding fragment heavy chain (24 kDa, Protein from Mus musculus)
Apo form of UIC2 Fab complex of human-mouse chimeric ABCB1 (ABCB1HM)
Resolution: 4.14 Å
EM Method: Single-particle
Fitted PDBs: 6fn4
Q-score: 0.34
Alam A, Kung R, Kowal J, McLeod RA, Tremp N, Broude EV, Roninson IB, Stahlberg H, Locher KP
PNAS (2018) 115 pp. E1973-E1982 [ DOI: doi:10.1073/pnas.1717044115 Pubmed: 29440498 ]
- Apo form of human-mouse chimeric abcb1 (abcb1hm) in complex with antigen binding fragment of uic2. (141 kDa, Protein from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- 1,2-distearoyl-sn-glycerophosphoethanolamine (748 Da, Ligand)
- Apo human-mouse chimeric abcb1 (abcb1hm) complex with uic2 fab (195 kDa, Complex)
- Uic2 antigen binding fragment light chain (24 kDa, Protein from Mus musculus)
- Apo human-mouse chimeric abcb1 (abcb1hm) complex with uic2 fab (142 kDa, Complex from Homo sapiens)
- Apo human-mouse chimeric abcb1 (abcb1hm) complex with uic2 fab (48 kDa, Complex from Mus musculus)
- Uic2 antigen binding fragment heavy chain (24 kDa, Protein from Mus musculus)
Apo form of UIC2 Fab complex of human-mouse chimeric ABCB1 (ABCB1HM) - Map 2 (kinked TM4 and TM10)
Alam A, Kung R, Kowal J, McLeod RA, Tremp N, Broude EV, Roninson IB, Stahlberg H, Locher KP
PNAS (2018) 115 pp. E1973-E1982 [ DOI: doi:10.1073/pnas.1717044115 Pubmed: 29440498 ]
- Apo human-mouse chimeric abcb1 (abcb1hm) complex with uic2 fab (195 kDa, Complex)
- Apo human-mouse chimeric abcb1 (abcb1hm) (142 kDa, Complex from Homo sapiens)
- Uic2 fab (48 kDa, Complex from Mus musculus)
Alam A, Kung R, Kowal J, McLeod RA, Tremp N, Broude EV, Roninson IB, Stahlberg H, Locher KP
PNAS (2018) 115 pp. E1973-E1982 [ DOI: doi:10.1073/pnas.1717044115 Pubmed: 29440498 ]
- Apo human-mouse chimeric abcb1 (abcb1hm) complex with uic2 fab (195 kDa, Complex)
- Apo human-mouse chimeric abcb1 (abcb1hm) (142 kDa, Complex from Homo sapiens)
- Uic2 fab (48 kDa, Complex from Mus musculus)
Alam A, Kung R, Kowal J, McLeod RA, Tremp N, Broude EV, Roninson IB, Stahlberg H, Locher KP
PNAS (2018) 115 pp. E1973-E1982 [ DOI: doi:10.1073/pnas.1717044115 Pubmed: 29440498 ]