Cryo-EM structure of H2DIDS-bound human Anion Exchanger 1
Capper MJ, Yang S, Stone AC, Vatansever S, Zilberg G, Mathiharan YK, Habib R, Hutchinson K, Zhao Y, Schlessinger A, Mezei M, Osman R, Zhang B, Wacker D
Nat Struct Mol Biol (2023) 30 pp. 1495-1504 [ Pubmed: 37679563 DOI: 10.1038/s41594-023-01085-6 ]
Image sets:
Cryo-EM structure of Bicarbonate-bound human Anion Exchanger 1
Capper MJ, Yang S, Stone AC, Vatansever S, Zilberg G, Mathiharan YK, Habib R, Hutchinson K, Zhao Y, Schlessinger A, Mezei M, Osman R, Zhang B, Wacker D
Nat Struct Mol Biol (2023) 30 pp. 1495-1504 [ Pubmed: 37679563 DOI: 10.1038/s41594-023-01085-6 ]
Image sets:
Cryo-EM structure of DIDS-bound human Anion Exchanger 1
Capper MJ, Yang S, Stone AC, Vatansever S, Zilberg G, Mathiharan YK, Habib R, Hutchinson K, Zhao Y, Schlessinger A, Mezei M, Osman R, Zhang B, Wacker D
Nat Struct Mol Biol (2023) 30 pp. 1495-1504 [ Pubmed: 37679563 DOI: 10.1038/s41594-023-01085-6 ]
Image sets:
Cryo-EM structure of Niflumic Acid-bound human Anion Exchanger 1
Capper MJ, Yang S, Stone AC, Vatansever S, Zilberg G, Mathiharan YK, Habib R, Hutchinson K, Zhao Y, Schlessinger A, Mezei M, Osman R, Zhang B, Wacker D
Nat Struct Mol Biol (2023) 30 pp. 1495-1504 [ Pubmed: 37679563 DOI: 10.1038/s41594-023-01085-6 ]
Image sets:
Cryo-EM structure of Dipyridamole-bound human Anion Exchanger 1
Capper MJ, Yang S, Stone AC, Vatansever S, Zilberg G, Mathiharan YK, Habib R, Hutchinson K, Zhao Y, Schlessinger A, Mezei M, Osman R, Zhang B, Wacker D
Nat Struct Mol Biol (2023) 30 pp. 1495-1504 [ Pubmed: 37679563 DOI: 10.1038/s41594-023-01085-6 ]
Image sets:
Cryo-EM structure of human Anion Exchanger 1 modified with Diethyl Pyrocarbonate (DEPC)
Capper MJ, Yang S, Stone AC, Vatansever S, Zilberg G, Mathiharan YK, Habib R, Hutchinson K, Zhao Y, Schlessinger A, Mezei M, Osman R, Zhang B, Wacker D
Nat Struct Mol Biol (2023) 30 pp. 1495-1504 [ Pubmed: 37679563 DOI: 10.1038/s41594-023-01085-6 ]
Image sets:
Cryo-EM structure of human Anion Exchanger 1
Capper MJ, Yang S, Stone AC, Vatansever S, Zilberg G, Mathiharan YK, Habib R, Hutchinson K, Zhao Y, Schlessinger A, Mezei M, Osman R, Zhang B, Wacker D
Nat Struct Mol Biol (2023) [ Pubmed: 37679563 DOI: 10.1038/s41594-023-01085-6 ]
Image sets:
Cryo-EM structure of human Anion Exchanger 1 bound to Dipyridamole
Resolution: 3.13 Å
EM Method: Single-particle
Fitted PDBs: 8t6u
Q-score: 0.469
Capper MJ, Yang S, Stone AC, Vatansever S, Zilberg G, Mathiharan YK, Habib R, Hutchinson K, Zhao Y, Schlessinger A, Mezei M, Osman R, Zhang B, Wacker D
Nat Struct Mol Biol (2023) 30 pp. 1495-1504 [ Pubmed: 37679563 DOI: doi:10.1038/s41594-023-01085-6 ]
- Water (18 Da, Ligand)
- Dimeric anion exchanger 1 (slc4a1) (203 kDa, Complex from Homo sapiens)
- 1,2-diacyl-sn-glycero-3-phosphocholine (790 Da, Ligand)
- Band 3 anion transport protein (58 kDa, Protein from Homo sapiens)
- 2-[[2-[bis(2-hydroxyethyl)amino]-4,8-di(piperidin-1-yl)pyrimido[5,4-d]pyrimidin-6-yl]-(2-hydroxyethyl)amino]ethanol (504 Da, Ligand)
- Cholesterol (386 Da, Ligand)
Resolution: 2.95 Å
EM Method: Single-particle
Fitted PDBs: 8t6v
Q-score: 0.479
Capper MJ, Yang S, Stone AC, Vatansever S, Zilberg G, Mathiharan YK, Habib R, Hutchinson K, Zhao Y, Schlessinger A, Mezei M, Osman R, Zhang B, Wacker D
Nat Struct Mol Biol (2023) 30 pp. 1495-1504 [ Pubmed: 37679563 DOI: doi:10.1038/s41594-023-01085-6 ]
- Water (18 Da, Ligand)
- Dimeric anion exchanger 1 (slc4a1) (203 kDa, Complex from Homo sapiens)
- Cholesterol hemisuccinate (486 Da, Ligand)
- 1,2-diacyl-sn-glycero-3-phosphocholine (790 Da, Ligand)
- 4,4'-diisothiocyano-2,2'-stilbenedisulfonic acid (454 Da, Ligand)
- Band 3 anion transport protein (58 kDa, Protein from Homo sapiens)
- Cholesterol (386 Da, Ligand)
Cryo-EM structure of human Anion Exchanger 1
Resolution: 2.99 Å
EM Method: Single-particle
Fitted PDBs: 7ty4
Q-score: 0.463
Capper MJ, Yang S, Stone AC, Vatansever S, Zilberg G, Mathiharan YK, Habib R, Hutchinson K, Zhao Y, Schlessinger A, Mezei M, Osman R, Zhang B, Wacker D
Nat Struct Mol Biol (2023) 30 pp. 1495-1504 [ Pubmed: 37679563 DOI: doi:10.1038/s41594-023-01085-6 ]
- Water (18 Da, Ligand)
- Dimeric anion exchanger 1 (slc4a1) (203 kDa, Complex from Homo sapiens)
- Cholesterol hemisuccinate (486 Da, Ligand)
- 1,2-diacyl-sn-glycero-3-phosphocholine (790 Da, Ligand)
- Band 3 anion transport protein (101 kDa, Protein from Homo sapiens)
- Cholesterol (386 Da, Ligand)