Nonactive state of Gly-,Glu- bound GluN1a-2B-2D NMDAR
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 Pubmed: 39954679 ]
- Tri-heteromeric glun1-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- Water (18 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glutamic acid (147 Da, Ligand)
- Glycine (75 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Open state of Gly-,Glu-,EU1622-240 bound GluN1a-2B-2D NMDAR
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 Pubmed: 39954679 ]
- Tri-heteromeric glun1-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glutamic acid (147 Da, Ligand)
- Glycine (75 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Gly-,PPDA- bound GluN1a-2B-2D NMDAR
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 Pubmed: 39954679 ]
- Tri-heteromeric glun1a-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- (2s,3r)-1-(phenanthren-2-ylcarbonyl)piperazine-2,3-dicarboxylic acid (378 Da, Ligand)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glycine (75 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Nonactive state of Gly-,Glu- bound GluN1a-2B-2D NMDAR (Low-res)
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 Pubmed: 39954679 ]
- Tri-heteromeric glun1-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glutamic acid (147 Da, Ligand)
- Glycine (75 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Gly-,Glu-,(S)-DQP-997-74 bound GluN1a-2B-2D NMDAR
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 Pubmed: 39954679 ]
- Tri-heteromeric glun1-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- 4-{(3r,5s)-5-(4-chlorophenyl)-3-[4-(4-chlorophenyl)-2-oxo-1,2-dihydroquinolin-3-yl]pyrazolidin-1-yl}-3,3-difluoro-4-oxobutanoic acid (572 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glutamic acid (147 Da, Ligand)
- Glycine (75 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Gly-,Glu-,(S)-(+)-ketamine bound GluN1a-2B-2D NMDAR
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 Pubmed: 39954679 ]
- Tri-heteromeric glun1-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- (2~{s})-2-(2-chlorophenyl)-2-(methylamino)cyclohexan-1-one (237 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glutamic acid (147 Da, Ligand)
- Glycine (75 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)