Nonactive state of Gly-,Glu- bound GluN1a-2B-2D NMDAR
Resolution: 3.34 Å
EM Method: Single-particle
Fitted PDBs: 9d37
Q-score: 0.443
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 ]
- Glutamic acid (147 Da, Ligand)
- Tri-heteromeric glun1-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glycine (75 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Water (18 Da, Ligand)
Open state of Gly-,Glu-,EU1622-240 bound GluN1a-2B-2D NMDAR
Resolution: 3.95 Å
EM Method: Single-particle
Fitted PDBs: 9d38
Q-score: 0.323
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 ]
- Glutamic acid (147 Da, Ligand)
- Tri-heteromeric glun1-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glycine (75 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Gly-,PPDA- bound GluN1a-2B-2D NMDAR
Resolution: 3.65 Å
EM Method: Single-particle
Fitted PDBs: 9d39
Q-score: 0.385
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 ]
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glycine (75 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- (2s,3r)-1-(phenanthren-2-ylcarbonyl)piperazine-2,3-dicarboxylic acid (378 Da, Ligand)
- Tri-heteromeric glun1a-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
Nonactive state of Gly-,Glu- bound GluN1a-2B-2D NMDAR (Low-res)
Resolution: 3.78 Å
EM Method: Single-particle
Fitted PDBs: 9d3a
Q-score: 0.368
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 ]
- Glutamic acid (147 Da, Ligand)
- Tri-heteromeric glun1-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glycine (75 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Gly-,Glu-,(S)-DQP-997-74 bound GluN1a-2B-2D NMDAR
Resolution: 3.71 Å
EM Method: Single-particle
Fitted PDBs: 9d3b
Q-score: 0.311
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 ]
- Glutamic acid (147 Da, Ligand)
- Tri-heteromeric glun1-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- 4-{(3r,5s)-5-(4-chlorophenyl)-3-[4-(4-chlorophenyl)-2-oxo-1,2-dihydroquinolin-3-yl]pyrazolidin-1-yl}-3,3-difluoro-4-oxobutanoic acid (572 Da, Ligand)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- Glycine (75 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Gly-,Glu-,(S)-(+)-ketamine bound GluN1a-2B-2D NMDAR
Resolution: 3.96 Å
EM Method: Single-particle
Fitted PDBs: 9d3c
Q-score: 0.353
Kang H, Epstein M, Banke TG, Perszyk R, Simorowski N, Paladugu S, Liotta DC, Traynelis SF, Furukawa H
Neuron (2025) [ DOI: doi:10.1016/j.neuron.2025.01.013 ]
- Glutamic acid (147 Da, Ligand)
- Tri-heteromeric glun1-2b-2d nmdar (377 kDa, Complex from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (94 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (92 kDa, Protein from Homo sapiens)
- (2~{s})-2-(2-chlorophenyl)-2-(methylamino)cyclohexan-1-one (237 Da, Ligand)
- Glycine (75 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2b (98 kDa, Protein from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
D-cycloserine and glutamate bound Human GluN1a-GluN2C NMDA receptor in intact conformation
Resolution: 3.96 Å
EM Method: Single-particle
Fitted PDBs: 8e92
Q-score: 0.397
Chou TH, Kang H, Simorowski N, Traynelis SF, Furukawa H
Mol Cell (2022) 82 pp. 4548- [ DOI: doi:10.1016/j.molcel.2022.10.008 Pubmed: 36309015 ]
- Glutamate receptor ionotropic, nmda 2c (96 kDa, Protein from Homo sapiens)
- Hetero-tetrameric glun1a-glun2c nmda receptors (Complex from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Glutamate receptor ionotropic, nmda 1 (95 kDa, Protein from Homo sapiens)
D-cycloserine and glutamate bound Human GluN1a-GluN2C NMDA receptor in splayed conformation
Resolution: 3.71 Å
EM Method: Single-particle
Fitted PDBs: 8e93
Q-score: 0.443
Chou TH, Kang H, Simorowski N, Traynelis SF, Furukawa H
Mol Cell (2022) 82 pp. 4548- [ DOI: doi:10.1016/j.molcel.2022.10.008 Pubmed: 36309015 ]
- Glutamate receptor ionotropic, nmda 2c (96 kDa, Protein from Homo sapiens)
- Hetero-tetrameric glun1a-glun2c nmda receptors (Complex from Homo sapiens)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Glutamate receptor ionotropic, nmda 1 (95 kDa, Protein from Homo sapiens)
PYD-106-bound Human GluN1a-GluN2C NMDA receptor in intact conformation
Resolution: 3.72 Å
EM Method: Single-particle
Fitted PDBs: 8e94
Q-score: 0.47
Chou TH, Kang H, Simorowski N, Traynelis SF, Furukawa H
Mol Cell (2022) 82 pp. 4548- [ DOI: doi:10.1016/j.molcel.2022.10.008 Pubmed: 36309015 ]
- Methyl 4-[(2~{r})-3-ethanoyl-1-[2-(2-methyl-1~{h}-indol-3-yl)ethyl]-4-oxidanyl-5-oxidanylidene-2~{h}-pyrrol-2-yl]benzoate (432 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Glutamate receptor ionotropic, nmda 2c (96 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 1 (95 kDa, Protein from Homo sapiens)
- Hetero-tetrameric glun1a-glun2c nmda receptors (Complex from Homo sapiens)
Glycine and glutamate bound Human GluN1a-GluN2D NMDA receptor
Resolution: 3.38 Å
EM Method: Single-particle
Fitted PDBs: 8e96
Q-score: 0.411
Chou TH, Kang H, Simorowski N, Traynelis SF, Furukawa H
Mol Cell (2022) 82 pp. 4548- [ DOI: doi:10.1016/j.molcel.2022.10.008 Pubmed: 36309015 ]
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Glutamate receptor ionotropic, nmda 1 (93 kDa, Protein from Homo sapiens)
- Glutamate receptor ionotropic, nmda 2d (96 kDa, Protein from Homo sapiens)
- Hetero-tetrameric glun1a-glun2d nmda receptors (Complex from Homo sapiens)
- Glutamic acid (147 Da, Ligand)
- Glycine (75 Da, Ligand)