Caenorhabditis elegans ACR-23 in betaine and monepantel bound state
Resolution: 2.64 Å
EM Method: Single-particle
Fitted PDBs: 8zfk
Q-score: 0.622
Liu F, Li T, Gong H, Tian F, Bai Y, Wang H, Yang C, Li Y, Guo F, Liu S, Chen Q
EMBO J (2024) 43 pp. 3787-3806 [ DOI: doi:10.1038/s44318-024-00165-7 Pubmed: 39009676 ]
- Water (18 Da, Ligand)
- ~{n}-[(2~{s})-2-cyano-1-[5-cyano-2-(trifluoromethyl)phenoxy]propan-2-yl]-4-(trifluoromethylsulfanyl)benzamide (473 Da, Ligand)
- Betaine receptor acr-23,soluble cytochrome b562 (70 kDa, Protein from Caenorhabditis elegans)
- Acetylcholine receptor like-23(acr-23) (67 kDa, Complex from Caenorhabditis elegans)
- Trimethyl glycine (118 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Caenorhabditis elegans ACR-23 in betaine bound state
Resolution: 2.96 Å
EM Method: Single-particle
Fitted PDBs: 8zfm
Q-score: 0.58
Liu F, Li T, Gong H, Tian F, Bai Y, Wang H, Yang C, Li Y, Guo F, Liu S, Chen Q
EMBO J (2024) 43 pp. 3787-3806 [ DOI: doi:10.1038/s44318-024-00165-7 Pubmed: 39009676 ]
- Trimethyl glycine (118 Da, Ligand)
- Acetylcholine receptor like-23(acr-23) (67 kDa, Complex from Caenorhabditis elegans)
- Water (18 Da, Ligand)
- Betaine receptor acr-23,soluble cytochrome b562 (70 kDa, Protein from Caenorhabditis elegans)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
Rat Kir4.1 in complex with PIP2
Resolution: 2.85 Å
EM Method: Single-particle
Fitted PDBs: 8i5m
Q-score: 0.486
Zhou X, Zhao C, Xu H, Xu Y, Zhan L, Wang P, He J, Lu T, Gu Y, Yang Y, Xu C, Chen Y, Liu Y, Zeng Y, Tian F, Chen Q, Xie X, Liu J, Hu H, Li J, Zheng Y, Guo J, Gao Z
Nat Chem Biol (2024) 20 pp. 857-866 [ Pubmed: 38355723 DOI: doi:10.1038/s41589-024-01555-y ]
- [(2r)-2-octanoyloxy-3-[oxidanyl-[(1r,2r,3s,4r,5r,6s)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate (746 Da, Ligand)
- Atp-sensitive inward rectifier potassium channel 10 (38 kDa, Protein from Rattus norvegicus)
- Rat kir4.1 in complex with pip2 (Complex from Rattus norvegicus)
Rat Kir4.1 in complex with PIP2 and Lys05
Resolution: 2.85 Å
EM Method: Single-particle
Fitted PDBs: 8i5n
Q-score: 0.414
Zhou X, Zhao C, Xu H, Xu Y, Zhan L, Wang P, He J, Lu T, Gu Y, Yang Y, Xu C, Chen Y, Liu Y, Zeng Y, Tian F, Chen Q, Xie X, Liu J, Hu H, Li J, Zheng Y, Guo J, Gao Z
Nat Chem Biol (2024) 20 pp. 857-866 [ Pubmed: 38355723 DOI: doi:10.1038/s41589-024-01555-y ]
- Rat kir4.1 in complex with pip2 and lys05 (Complex from Rattus norvegicus)
- Atp-sensitive inward rectifier potassium channel 10 (38 kDa, Protein from Rattus norvegicus)
- [(2r)-2-octanoyloxy-3-[oxidanyl-[(1r,2r,3s,4r,5r,6s)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate (746 Da, Ligand)