Rabbit Cav1.1-Nifedipine Complex
Resolution: 2.9 Å
EM Method: Single-particle
Fitted PDBs: 6jp5
Q-score: 0.39
Zhao Y, Huang G, Wu J, Wu Q, Gao S, Yan Z, Lei J, Yan N
Cell (2019) 177 pp. 1495-1506.e12 [ DOI: doi:10.1016/j.cell.2019.04.043 Pubmed: 31150622 ]
- Voltage-dependent l-type calcium channel subunit beta-1 (49 kDa, Protein from Oryctolagus cuniculus)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Calcium ion (40 Da, Ligand)
- 1,2-distearoyl-sn-glycerophosphoethanolamine (748 Da, Ligand)
- 1,2-diacyl-sn-glycero-3-phosphocholine (790 Da, Ligand)
- Dimethyl 2,6-dimethyl-4-(2-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate (346 Da, Ligand)
- Voltage-dependent calcium channel subunit alpha-2/delta-1 (121 kDa, Protein from Oryctolagus cuniculus)
- Cav1.1-drug complex (Complex)
- Cav1.1-beta1a-alpha2-delta1-gamma complex (Complex from Oryctolagus cuniculus)
- Voltage-dependent l-type calcium channel subunit alpha-1s (212 kDa, Protein from Oryctolagus cuniculus)
- Ethanolamine (61 Da, Ligand)
- Voltage-dependent calcium channel gamma-1 subunit (25 kDa, Protein from Oryctolagus cuniculus)
Rabbit Cav1.1-Bay K8644 Complex
Resolution: 2.7 Å
EM Method: Single-particle
Fitted PDBs: 6jp8
Q-score: 0.385
Zhao Y, Huang G, Wu J, Wu Q, Gao S, Yan Z, Lei J, Yan N
Cell (2019) 177 pp. 1495-1506.e12 [ DOI: doi:10.1016/j.cell.2019.04.043 Pubmed: 31150622 ]
- Voltage-dependent l-type calcium channel subunit beta-1 (49 kDa, Protein from Oryctolagus cuniculus)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Calcium ion (40 Da, Ligand)
- Voltage-dependent calcium channel subunit alpha-2/delta-1 (118 kDa, Protein from Oryctolagus cuniculus)
- Cav1.1-drug complex (Complex)
- Methyl (4~{s})-2,6-dimethyl-5-nitro-4-[2-(trifluoromethyl)phenyl]-1,4-dihydropyridine-3-carboxylate (356 Da, Ligand)
- Cav1.1-beta1a-alpha2-delta1-gamma complex (Complex from Oryctolagus cuniculus)
- Voltage-dependent l-type calcium channel subunit alpha-1s (212 kDa, Protein from Oryctolagus cuniculus)
- Ethanolamine (61 Da, Ligand)
- Voltage-dependent calcium channel gamma-1 subunit (25 kDa, Protein from Oryctolagus cuniculus)
Rabbit Cav1.1-Verapamil Complex
Resolution: 2.6 Å
EM Method: Single-particle
Fitted PDBs: 6jpa
Q-score: 0.4
Zhao Y, Huang G, Wu J, Wu Q, Gao S, Yan Z, Lei J, Yan N
Cell (2019) 177 pp. 1495-1506.e12 [ DOI: doi:10.1016/j.cell.2019.04.043 Pubmed: 31150622 ]
- Voltage-dependent l-type calcium channel subunit beta-1 (49 kDa, Protein from Oryctolagus cuniculus)
- Voltage-dependent l-type calcium channel subunit beta-1 (57 kDa, Protein from Oryctolagus cuniculus)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Calcium ion (40 Da, Ligand)
- 1,2-distearoyl-sn-glycerophosphoethanolamine (748 Da, Ligand)
- Voltage-dependent calcium channel subunit alpha-2/delta-1 (118 kDa, Protein from Oryctolagus cuniculus)
- 1,2-diacyl-sn-glycero-3-phosphocholine (790 Da, Ligand)
- (3beta,14beta,17beta,25r)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en (544 Da, Ligand)
- Cav1.1-drug complex (Complex)
- (2s)-2-(3,4-dimethoxyphenyl)-5-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}-2-(propan-2-yl)pentanenitrile (454 Da, Ligand)
- Cav1.1-beta1a-alpha2-delta1-gamma complex (Complex from Oryctolagus cuniculus)
- Ethanolamine (61 Da, Ligand)
- Voltage-dependent calcium channel gamma-1 subunit (25 kDa, Protein from Oryctolagus cuniculus)
- Voltage-dependent l-type calcium channel subunit alpha-1s (172 kDa, Protein from Oryctolagus cuniculus)
Rabbit Cav1.1-Diltiazem Complex
Resolution: 2.9 Å
EM Method: Single-particle
Fitted PDBs: 6jpb
Q-score: 0.397
Zhao Y, Huang G, Wu J, Wu Q, Gao S, Yan Z, Lei J, Yan N
Cell (2019) 177 pp. 1495-1506.e12 [ DOI: doi:10.1016/j.cell.2019.04.043 Pubmed: 31150622 ]
- Voltage-dependent l-type calcium channel subunit beta-1 (49 kDa, Protein from Oryctolagus cuniculus)
- Diltiazem (414 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Calcium ion (40 Da, Ligand)
- 1,2-distearoyl-sn-glycerophosphoethanolamine (748 Da, Ligand)
- 1,2-diacyl-sn-glycero-3-phosphocholine (790 Da, Ligand)
- Voltage-dependent calcium channel subunit alpha-2/delta-1 (118 kDa, Protein from Oryctolagus cuniculus)
- Cav1.1-drug complex (Complex)
- Cav1.1-beta1a-alpha2-delta1-gamma complex (Complex from Oryctolagus cuniculus)
- Voltage-dependent l-type calcium channel subunit alpha-1s (212 kDa, Protein from Oryctolagus cuniculus)
- Ethanolamine (61 Da, Ligand)
- Voltage-dependent calcium channel gamma-1 subunit (25 kDa, Protein from Oryctolagus cuniculus)
- Voltage-dependent l-type calcium channel subunit beta-1 (57 kDa, Protein from Oryctolagus cuniculus)