CXCR3-DNGi complex activated by CXCL11
Resolution: 3.01 Å
EM Method: Single-particle
Fitted PDBs: 8hnk
Q-score: 0.532
Jiao H, Pang B, Liu A, Chen Q, Pan Q, Wang X, Xu Y, Chiang YC, Ren R, Hu H
Nat Struct Mol Biol (2024) 31 pp. 610-620 [ Pubmed: 38177682 DOI: doi:10.1038/s41594-023-01175-5 ]
- C-x-c motif chemokine 11 (11 kDa, Protein from Homo sapiens)
- Cholesterol (386 Da, Ligand)
- Guanine nucleotide-binding protein g(i) subunit alpha-1 (40 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (42 kDa, Protein from Homo sapiens)
- Single-chain variable fragment scfv16 (27 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Homo sapiens)
- Soluble cytochrome b562,c-x-c chemokine receptor type 3,oplophorus-luciferin 2-monooxygenase catalytic subunit (72 kDa, Protein from Oplophorus gracilirostris)
- Cxcr3-cxcl11-dngi-scfv16 (Complex from Homo sapiens)
CXCR3-DNGi complex activated by PS372424
Resolution: 2.98 Å
EM Method: Single-particle
Fitted PDBs: 8hnl
Q-score: 0.548
Jiao H, Pang B, Liu A, Chen Q, Pan Q, Wang X, Xu Y, Chiang YC, Ren R, Hu H
Nat Struct Mol Biol (2024) 31 pp. 610-620 [ DOI: doi:10.1038/s41594-023-01175-5 Pubmed: 38177682 ]
- Single-chain variable fragment scfv16 (27 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Homo sapiens)
- (3s)-n-[(2s)-5-carbamimidamido-1-(cyclohexylmethylamino)-1-oxidanylidene-pentan-2-yl]-2-(4-oxidanylidene-4-phenyl-butanoyl)-3,4-dihydro-1h-isoquinoline-3-carboxamide (588 Da, Ligand)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (42 kDa, Protein from Homo sapiens)
- Cxcr3-ps372424-dngi-scfv16 (Complex from Homo sapiens)
- Guanine nucleotide-binding protein g(i) subunit alpha-1 (40 kDa, Protein from Homo sapiens)
- Cholesterol (386 Da, Ligand)
- Soluble cytochrome b562,c-x-c chemokine receptor type 3,oplophorus-luciferin 2-monooxygenase catalytic subunit (72 kDa, Protein from Oplophorus gracilirostris)
CXCR3-DNGi complex activated by VUF11222
Resolution: 2.94 Å
EM Method: Single-particle
Fitted PDBs: 8hnm
Q-score: 0.546
Jiao H, Pang B, Liu A, Chen Q, Pan Q, Wang X, Xu Y, Chiang YC, Ren R, Hu H
Nat Struct Mol Biol (2024) 31 pp. 610-620 [ DOI: doi:10.1038/s41594-023-01175-5 Pubmed: 38177682 ]
- Single-chain variable fragment scfv16 (27 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (7 kDa, Protein from Homo sapiens)
- [4-(2-bromophenyl)phenyl]methyl-[[(1r,5s)-6,6-dimethyl-2-bicyclo[3.1.1]hept-2-enyl]methyl]-dimethyl-azanium (425 Da, Ligand)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (42 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i) subunit alpha-1 (40 kDa, Protein from Homo sapiens)
- Cxcr3-vuf11222-dngi-scfv16 (Complex from Homo sapiens)
- Cholesterol (386 Da, Ligand)
- Soluble cytochrome b562,c-x-c chemokine receptor type 3,oplophorus-luciferin 2-monooxygenase catalytic subunit (72 kDa, Protein from Oplophorus gracilirostris)