mouse proteasome 20S subunit in complex with compound 1
Resolution: 2.7 Å
EM Method: Single-particle
Fitted PDBs: 8ypk
Q-score: 0.621
Arai Y, Shitama H, Yamagishi M, Ono S, Kashima A, Hiraizumi M, Tsuda N, Katayama K, Tanaka K, Koda Y, Kato S, Sakata K, Nureki O, Miyazaki H
Bioorg.Med.Chem. (2024) 109 pp. 117790-117790 [ Pubmed: 38906067 DOI: doi:10.1016/j.bmc.2024.117790 ]
- Proteasome subunit alpha type-1 (29 kDa, Protein from Mus musculus)
- Proteasome subunit alpha type-2 (25 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-2 (22 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-7 (25 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-6 (22 kDa, Protein from Mus musculus)
- Proteasome subunit alpha type-6 (27 kDa, Protein from Mus musculus)
- [(1r)-1-[(1-cyclohexyl-1,2,3-triazol-4-yl)carbonylamino]-3-methyl-butyl]boronic acid (308 Da, Ligand)
- Proteasome subunit alpha type-4 (29 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-5 (22 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-4 (29 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-3 (22 kDa, Protein from Mus musculus)
- Proteasome subunit alpha type-3 (28 kDa, Protein from Mus musculus)
- 20s proteasome (Complex from Mus musculus)
- Proteasome subunit alpha type-5 (26 kDa, Protein from Mus musculus)
- Proteasome subunit alpha type-7 (27 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-1 (26 kDa, Protein from Mus musculus)
canine immunoproteasome 20S subunit in complex with compound 2
Resolution: 2.2 Å
EM Method: Single-particle
Fitted PDBs: 8ysx
Q-score: 0.541
Arai Y, Shitama H, Yamagishi M, Ono S, Kashima A, Hiraizumi M, Tsuda N, Katayama K, Tanaka K, Koda Y, Kato S, Sakata K, Nureki O, Miyazaki H
Bioorg.Med.Chem. (2024) 109 pp. 117790-117790 [ Pubmed: 38906067 DOI: doi:10.1016/j.bmc.2024.117790 ]
- Proteasome subunit alpha type (26 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit alpha type (27 kDa, Protein from Canis lupus familiaris)
- Water (18 Da, Ligand)
- [(~{r})-cyclohexyl-[(1-cyclohexyl-1,2,3-triazol-4-yl)carbonylamino]methyl]boronic acid (334 Da, Ligand)
- Proteasome subunit alpha type (25 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit alpha type (29 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (22 kDa, Protein from Canis lupus familiaris)
- 20s immunoproteasome (Complex from Canis lupus familiaris)
- Proteasome subunit alpha type (29 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (23 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit alpha type (27 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (29 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (24 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (26 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (21 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta type-8 (22 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit alpha type (28 kDa, Protein from Canis lupus familiaris)
canine immunoproteasome 20S subunit in complex with compound 1
Resolution: 2.0 Å
EM Method: Single-particle
Fitted PDBs: 8yvg
Q-score: 0.707
Arai Y, Shitama H, Yamagishi M, Ono S, Kashima A, Hiraizumi M, Tsuda N, Katayama K, Tanaka K, Koda Y, Kato S, Sakata K, Nureki O, Miyazaki H
Bioorg.Med.Chem. (2024) 109 pp. 117790-117790 [ Pubmed: 38906067 DOI: doi:10.1016/j.bmc.2024.117790 ]
- Proteasome subunit alpha type (26 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit alpha type (27 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (26 kDa, Protein from Canis lupus familiaris)
- [(1r)-1-[(1-cyclohexyl-1,2,3-triazol-4-yl)carbonylamino]-3-methyl-butyl]boronic acid (308 Da, Ligand)
- Proteasome subunit alpha type (25 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (22 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit alpha type (29 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit alpha type (29 kDa, Protein from Canis lupus familiaris)
- 20s immunoproteasome (Complex from Canis lupus familiaris)
- Proteasome subunit beta (23 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit alpha type (27 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (29 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit alpha type (28 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (21 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta type-8 (22 kDa, Protein from Canis lupus familiaris)
- Proteasome subunit beta (29 kDa, Protein from Canis lupus familiaris)
canine immunoproteasome 20S subunit in complex with compound 1
Resolution: 2.5 Å
EM Method: Single-particle
Fitted PDBs: 8yvp
Q-score: 0.64
Arai Y, Shitama H, Yamagishi M, Ono S, Kashima A, Hiraizumi M, Tsuda N, Katayama K, Tanaka K, Koda Y, Kato S, Sakata K, Nureki O, Miyazaki H
Bioorg.Med.Chem. (2024) 109 pp. 117790-117790 [ Pubmed: 38906067 DOI: doi:10.1016/j.bmc.2024.117790 ]
- Proteasome subunit alpha type-1 (29 kDa, Protein from Mus musculus)
- Proteasome subunit alpha type-2 (25 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-2 (22 kDa, Protein from Mus musculus)
- [(~{r})-cyclohexyl-[(1-cyclohexyl-1,2,3-triazol-4-yl)carbonylamino]methyl]boronic acid (334 Da, Ligand)
- Proteasome subunit beta type-7 (25 kDa, Protein from Mus musculus)
- Proteasome subunit alpha type-6 (27 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-6 (22 kDa, Protein from Mus musculus)
- Proteasome subunit alpha type-4 (29 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-5 (22 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-3 (22 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-4 (29 kDa, Protein from Mus musculus)
- Proteasome subunit alpha type-3 (28 kDa, Protein from Mus musculus)
- 20s proteasome (Complex from Mus musculus)
- Proteasome subunit alpha type-5 (26 kDa, Protein from Mus musculus)
- Proteasome subunit alpha type-7 (27 kDa, Protein from Mus musculus)
- Proteasome subunit beta type-1 (26 kDa, Protein from Mus musculus)
- Threonine (119 Da, Ligand)