Oh S, Lee J, Choi HJ, Kim S, Sapuru V, Kim M, Hite RK
J Am Chem Soc (2024) 146 pp. 23230-23239 [ Pubmed: 39116214 DOI: doi:10.1021/jacs.4c05623 ]
- (2p,2'p)-2,2'-(1,3-phenylene)di(pyridin-4-amine) (262 Da, Ligand)
- Human tmem175 in an inhibitor-bound state (55 MDa, Complex from Homo sapiens)
- Endosomal/lysosomal potassium channel tmem175 (55 kDa, Protein from Homo sapiens)
Human Type 3 IP3 Receptor - Resting State (+IP3/ATP)
Resolution: 2.7 Å
EM Method: Single-particle
Fitted PDBs: 8tk8
Q-score: 0.524
Nat Commun (2023) 14 pp. 6897-6897 [ Pubmed: 37898605 DOI: doi:10.1038/s41467-023-42707-3 ]
- Inositol 1,4,5-trisphosphate receptor type 3 (304 kDa, Protein from Homo sapiens)
- Adenosine-5'-triphosphate (507 Da, Ligand)
- Zinc ion (65 Da, Ligand)
- 1,2-dioleoyl-sn-glycero-3-phosphocholine (787 Da, Ligand)
- Human type 3 ip3 receptor (1 MDa, Complex from Homo sapiens)
- D-myo-inositol-1,4,5-triphosphate (420 Da, Ligand)
Human Type 3 IP3 Receptor - 3:1 Resting-to-Preactivated Transition State
Nat Commun (2023) 14 pp. 6897-6897 [ Pubmed: 37898605 DOI: doi:10.1038/s41467-023-42707-3 ]
- Human type 3 ip3 receptor (1 MDa, Complex from Homo sapiens)
- Human type 3 ip3 receptor (Protein from Homo sapiens)
Human Type 3 IP3 Receptor - 2:2 Resting-to-Preactivated Transition State
Nat Commun (2023) 14 pp. 6897-6897 [ Pubmed: 37898605 DOI: doi:10.1038/s41467-023-42707-3 ]
- Human type 3 ip3 receptor (1 MDa, Complex from Homo sapiens)
- Human type 3 ip3 receptor (Protein from Homo sapiens)
Human Type 3 IP3 Receptor - 1:3 Resting-to-Preactivated Transition State
Nat Commun (2023) 14 pp. 6897-6897 [ Pubmed: 37898605 DOI: doi:10.1038/s41467-023-42707-3 ]
- Human type 3 ip3 receptor (1 MDa, Complex from Homo sapiens)
- Human type 3 ip3 receptor (Protein from Homo sapiens)
Human Type 3 IP3 Receptor - ARM2 Retraction Figure 4B
Nat Commun (2023) 14 pp. 6897-6897 [ Pubmed: 37898605 DOI: doi:10.1038/s41467-023-42707-3 ]
- Human type 3 ip3 receptor (1 MDa, Complex from Homo sapiens)
- Human type 3 ip3 receptor (Protein from Homo sapiens)
Human Type 3 IP3 Receptor - ARM2 Retraction Figure 4C
Nat Commun (2023) 14 pp. 6897-6897 [ Pubmed: 37898605 DOI: doi:10.1038/s41467-023-42707-3 ]
- Human type 3 ip3 receptor (1 MDa, Complex from Homo sapiens)
- Human type 3 ip3 receptor (Protein from Homo sapiens)
Human Type 3 IP3 Receptor - ARM2 Retraction Figure 4D
Nat Commun (2023) 14 pp. 6897-6897 [ Pubmed: 37898605 DOI: doi:10.1038/s41467-023-42707-3 ]
- Human type 3 ip3 receptor (1 MDa, Complex from Homo sapiens)
- Human type 3 ip3 receptor (Protein from Homo sapiens)
Human Type 3 IP3 Receptor - ARM2 Retraction Figure 4E
Nat Commun (2023) 14 pp. 6897-6897 [ Pubmed: 37898605 DOI: doi:10.1038/s41467-023-42707-3 ]
- Human type 3 ip3 receptor (1 MDa, Complex from Homo sapiens)
- Human type 3 ip3 receptor (Protein from Homo sapiens)
Human Type 3 IP3 Receptor - ARM2 Retraction Figure 4F
Nat Commun (2023) 14 pp. 6897-6897 [ Pubmed: 37898605 DOI: doi:10.1038/s41467-023-42707-3 ]
- Human type 3 ip3 receptor (1 MDa, Complex from Homo sapiens)
- Human type 3 ip3 receptor (Protein from Homo sapiens)