Cryo-EM structure of inhibitor 25a bound human urea transporter A2.
Resolution: 2.6 Å
EM Method: Single-particle
Fitted PDBs: 8xd7
Q-score: 0.461
Huang SM, Huang ZZ, Liu L, Xiong MY, Zhang C, Cai BY, Wang MW, Cai K, Jia YL, Wang JL, Zhang MH, Xie YH, Li M, Zhang H, Weng CH, Wen X, Li Z, Sun Y, Yi F, Yang Z, Xiao P, Yang F, Yu X, Tie L, Yang BX, Sun JP
Nat Commun (2024) 15 pp. 10226-10226 [ Pubmed: 39587082 DOI: doi:10.1038/s41467-024-54305-y ]
Cryo-EM structure of human urea transporter A2.
Resolution: 2.8 Å
EM Method: Single-particle
Fitted PDBs: 8xd9
Q-score: 0.547
Huang SM, Huang ZZ, Liu L, Xiong MY, Zhang C, Cai BY, Wang MW, Cai K, Jia YL, Wang JL, Zhang MH, Xie YH, Li M, Zhang H, Weng CH, Wen X, Li Z, Sun Y, Yi F, Yang Z, Xiao P, Yang F, Yu X, Tie L, Yang BX, Sun JP
Nat Commun (2024) 15 pp. 10226-10226 [ Pubmed: 39587082 DOI: doi:10.1038/s41467-024-54305-y ]
- Homotrimer complex of human urea transporter (Complex from Homo sapiens)
- Urea transporter 2 (43 kDa, Protein from Homo sapiens)
Cryo-EM structure of urea bound human urea transporter A2.
Resolution: 3.0 Å
EM Method: Single-particle
Fitted PDBs: 8xda
Q-score: 0.54
Huang SM, Huang ZZ, Liu L, Xiong MY, Zhang C, Cai BY, Wang MW, Cai K, Jia YL, Wang JL, Zhang MH, Xie YH, Li M, Zhang H, Weng CH, Wen X, Li Z, Sun Y, Yi F, Yang Z, Xiao P, Yang F, Yu X, Tie L, Yang BX, Sun JP
Nat Commun (2024) 15 pp. 10226-10226 [ Pubmed: 39587082 DOI: doi:10.1038/s41467-024-54305-y ]
- Homotrimer complex of human urea transporter (Complex from Homo sapiens)
- Urea (60 Da, Ligand)
- Water (18 Da, Ligand)
- Urea transporter 2 (43 kDa, Protein from Homo sapiens)
Cryo-EM structure of human urea transporter A2.
Resolution: 3.3 Å
EM Method: Single-particle
Fitted PDBs: 8xdb
Q-score: 0.515
Huang SM, Huang ZZ, Liu L, Xiong MY, Zhang C, Cai BY, Wang MW, Cai K, Jia YL, Wang JL, Zhang MH, Xie YH, Li M, Zhang H, Weng CH, Wen X, Li Z, Sun Y, Yi F, Yang Z, Xiao P, Yang F, Yu X, Tie L, Yang BX, Sun JP
Nat Commun (2024) 15 pp. 10226-10226 [ Pubmed: 39587082 DOI: doi:10.1038/s41467-024-54305-y ]
Cryo-EM structure of human urea transporter A2.
Resolution: 3.0 Å
EM Method: Single-particle
Fitted PDBs: 8xdc
Q-score: 0.562
Huang SM, Huang ZZ, Liu L, Xiong MY, Zhang C, Cai BY, Wang MW, Cai K, Jia YL, Wang JL, Zhang MH, Xie YH, Li M, Zhang H, Weng CH, Wen X, Li Z, Sun Y, Yi F, Yang Z, Xiao P, Yang F, Yu X, Tie L, Yang BX, Sun JP
Nat Commun (2024) 15 pp. 10226-10226 [ Pubmed: 39587082 DOI: doi:10.1038/s41467-024-54305-y ]
Cryo-EM structure of human urea transporter A2.
Resolution: 3.0 Å
EM Method: Single-particle
Fitted PDBs: 8xdd
Q-score: 0.524
Huang SM, Huang ZZ, Liu L, Xiong MY, Zhang C, Cai BY, Wang MW, Cai K, Jia YL, Wang JL, Zhang MH, Xie YH, Li M, Zhang H, Weng CH, Wen X, Li Z, Sun Y, Yi F, Yang Z, Xiao P, Yang F, Yu X, Tie L, Yang BX, Sun JP
Nat Commun (2024) 15 pp. 10226-10226 [ Pubmed: 39587082 DOI: doi:10.1038/s41467-024-54305-y ]
- Homotrimer complex of human urea transporter (Complex from Homo sapiens)
- 8-hydroxyquinoline-2-carboxylic acid (189 Da, Ligand)
- Urea transporter 2 (43 kDa, Protein from Homo sapien)
- 1-(3-methoxyphenyl)methanamine (137 Da, Ligand)
Cryo-EM structure of human urea transporter A3.
Resolution: 2.3 Å
EM Method: Single-particle
Fitted PDBs: 8xde
Q-score: 0.638
Huang SM, Huang ZZ, Liu L, Xiong MY, Zhang C, Cai BY, Wang MW, Cai K, Jia YL, Wang JL, Zhang MH, Xie YH, Li M, Zhang H, Weng CH, Wen X, Li Z, Sun Y, Yi F, Yang Z, Xiao P, Yang F, Yu X, Tie L, Yang BX, Sun JP
Nat Commun (2024) 15 pp. 10226-10226 [ Pubmed: 39587082 DOI: doi:10.1038/s41467-024-54305-y ]
- Homotrimer complex of human urea transporter (Complex from Homo sapiens)
- Urea transporter 2 (49 kDa, Protein from Homo sapiens)
Transporter associated with antigen processing (TAP) bound to the 9-mer peptide ILKEPVHGV
Resolution: 3.5 Å
EM Method: Single-particle
Fitted PDBs: 8t4e
Q-score: 0.438
Lee J, Oldham ML, Manon V, Chen J
PNAS (2024) 121 pp. e2320879121-e2320879121 [ Pubmed: 38805290 DOI: doi:10.1073/pnas.2320879121 ]
- Antigen peptide transporter 1 (81 kDa, Protein from Homo sapiens)
- Transframe peptide (993 Da, Protein from Human immunodeficiency virus 1)
- Transporter associated with antigen processing bound to the 9-mer peptide ilkepvhgv (156 kDa, Complex from Homo sapiens)
- Antigen peptide transporter 2 (75 kDa, Protein from Homo sapiens)
Transporter associated with antigen processing (TAP) bound to the 9-mer peptide RRYQKSTEL
Resolution: 3.5 Å
EM Method: Single-particle
Fitted PDBs: 8t4f
Q-score: 0.459
Lee J, Oldham ML, Manon V, Chen J
PNAS (2024) 121 pp. e2320879121-e2320879121 [ Pubmed: 38805290 DOI: doi:10.1073/pnas.2320879121 ]
- Antigen peptide transporter 1 (81 kDa, Protein from Homo sapiens)
- Antigen peptide transporter 2 (75 kDa, Protein from Homo sapiens)
- Transporter associated with antigen processing bound to the 9-mer peptide rryqkstel (156 kDa, Complex from Homo sapiens)
- Histone h3.3c peptide (1 kDa, Protein from Homo sapiens)
Transporter associated with antigen processing (TAP) bound to the 9-mer peptide QYDDAVYKL
Resolution: 3.5 Å
EM Method: Single-particle
Fitted PDBs: 8t4g
Q-score: 0.459
Lee J, Oldham ML, Manon V, Chen J
PNAS (2024) 121 pp. e2320879121-e2320879121 [ Pubmed: 38805290 DOI: doi:10.1073/pnas.2320879121 ]
- Transporter associated with antigen processing bound to the 9-mer peptide qyddavykl (156 kDa, Complex from Homo sapiens)
- Hla-c4 specific peptide (1 kDa, Protein from synthetic construct)
- Antigen peptide transporter 2 (75 kDa, Protein from Homo sapiens)
- Antigen peptide transporter 1 (81 kDa, Protein from Homo sapiens)