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- Autocatalytic activation of the furin zymogen requires removal of the emerging enzyme's N-terminus from the active site. Gawlik K, Shiryaev SA, Zhu W, Motamedchaboki K, Desjardins R, Day R, Remacle AG, Stec B, Strongin AY. PLoS ONE 4 e5031 (2009)
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- A novel enediynyl peptide inhibitor of furin that blocks processing of proPDGF-A, B and proVEGF-C. Basak A, Khatib AM, Mohottalage D, Basak S, Kolajova M, Bag SS, Basak A. PLoS ONE 4 e7700 (2009)
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- Structure of the unliganded form of the proprotein convertase furin suggests activation by a substrate-induced mechanism. Dahms SO, Arciniega M, Steinmetzer T, Huber R, Than ME. Proc. Natl. Acad. Sci. U.S.A. 113 11196-11201 (2016)
- Proprotein convertase subtilisin/kexin type 7 (PCSK7) is essential for the zebrafish development and bioavailability of transforming growth factor β1a (TGFβ1a). Turpeinen H, Oksanen A, Kivinen V, Kukkurainen S, Uusimäki A, Rämet M, Parikka M, Hytönen VP, Nykter M, Pesu M. J. Biol. Chem. 288 36610-36623 (2013)
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- Differential recognition of Old World and New World arenavirus envelope glycoproteins by subtilisin kexin isozyme 1 (SKI-1)/site 1 protease (S1P). Burri DJ, da Palma JR, Seidah NG, Zanotti G, Cendron L, Pasquato A, Kunz S. J. Virol. 87 6406-6414 (2013)
- Structural basis for dual-inhibition mechanism of a non-classical Kazal-type serine protease inhibitor from horseshoe crab in complex with subtilisin. Shenoy RT, Thangamani S, Velazquez-Campoy A, Ho B, Ding JL, Sivaraman J. PLoS ONE 6 e18838 (2011)
- Structure of Furin Protease Binding to SARS-CoV-2 Spike Glycoprotein and Implications for Potential Targets and Virulence. Vankadari N. J Phys Chem Lett 11 6655-6663 (2020)
- Identification of serpin determinants of specificity and selectivity for furin inhibition through studies of α1PDX (α1-protease inhibitor Portland)-serpin B8 and furin active-site loop chimeras. Izaguirre G, Qi L, Lima M, Olson ST. J. Biol. Chem. 288 21802-21814 (2013)
- Crystal structure of inhibitor-bound human MSPL that can activate high pathogenic avian influenza. Ohno A, Maita N, Tabata T, Nagano H, Arita K, Ariyoshi M, Uchida T, Nakao R, Ulla A, Sugiura K, Kishimoto K, Teshima-Kondo S, Okumura Y, Nikawa T. Life Sci Alliance 4 e202000849 (2021)
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