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- Design and synthesis of novel benzimidazole derivatives as phosphodiesterase 10A inhibitors with reduced CYP1A2 inhibition. Hamaguchi W, Masuda N, Isomura M, Miyamoto S, Kikuchi S, Amano Y, Honbou K, Mihara T, Watanabe T. Bioorg Med Chem 21 7612-7623 (2013)
- Synthesis of Fluorine-Containing Phosphodiesterase 10A (PDE10A) Inhibitors and the In Vivo Evaluation of F-18 Labeled PDE10A PET Tracers in Rodent and Nonhuman Primate. Li J, Zhang X, Jin H, Fan J, Flores H, Perlmutter JS, Tu Z. J Med Chem 58 8584-8600 (2015)
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- Novel benzimidazole derivatives as phosphodiesterase 10A (PDE10A) inhibitors with improved metabolic stability. Chino A, Masuda N, Amano Y, Honbou K, Mihara T, Yamazaki M, Tomishima M. Bioorg Med Chem 22 3515-3526 (2014)
- Synthesis, SAR study, and biological evaluation of novel quinoline derivatives as phosphodiesterase 10A inhibitors with reduced CYP3A4 inhibition. Hamaguchi W, Masuda N, Miyamoto S, Shiina Y, Kikuchi S, Mihara T, Moriguchi H, Fushiki H, Murakami Y, Amano Y, Honbou K, Hattori K. Bioorg Med Chem 23 297-313 (2015)
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- Addressing phototoxicity observed in a novel series of biaryl derivatives: discovery of potent, selective and orally active phosphodiesterase 10A inhibitor ASP9436. Hamaguchi W, Masuda N, Miyamoto S, Kikuchi S, Narazaki F, Shiina Y, Seo R, Amano Y, Mihara T, Moriguchi H, Hattori K. Bioorg Med Chem 23 3351-3367 (2015)
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- Inhibition mechanism exploration of quinoline derivatives as PDE10A inhibitors by in silico analysis. Wu Q, Gao Q, Guo H, Li D, Wang J, Gao W, Han C, Li Y, Yang L. Mol Biosyst 9 386-397 (2013)
- Design and optimization of purine derivatives as in vivo active PDE10A inhibitors. Chen L, Chen D, Tang L, Ren J, Chen J, Zhen X, Liu YC, Zhang C, Luo H, Shen J, Xiong B. Bioorg Med Chem 25 3315-3329 (2017)