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- Pharmaceutical and medicinal significance of sulfur (SVI)-Containing motifs for drug discovery: A critical review. Zhao C, Rakesh KP, Ravidar L, Fang WY, Qin HL. Eur J Med Chem 162 679-734 (2019)
- Chalcone and its analogs: Therapeutic and diagnostic applications in Alzheimer's disease. Thapa P, Upadhyay SP, Suo WZ, Singh V, Gurung P, Lee ES, Sharma R, Sharma M. Bioorg Chem 108 104681 (2021)
- Ghrelin octanoylation by ghrelin O-acyltransferase: protein acylation impacting metabolic and neuroendocrine signalling. Davis TR, Pierce MR, Novak SX, Hougland JL. Open Biol 11 210080 (2021)
- Recent Progress on Biological Activity of Amaryllidaceae and Further Isoquinoline Alkaloids in Connection with Alzheimer's Disease. Cahlíková L, Vrabec R, Pidaný F, Peřinová R, Maafi N, Mamun AA, Ritomská A, Wijaya V, Blunden G. Molecules 26 5240 (2021)
- An Overview of 1,2,3-triazole-Containing Hybrids and Their Potential Anticholinesterase Activities. Khan SA, Akhtar MJ, Gogoi U, Meenakshi DU, Das A. Pharmaceuticals (Basel) 16 179 (2023)
- Computer Aided Drug Design Methodologies with Natural Products in the Drug Research Against Alzheimer's Disease. de Sousa NF, Scotti L, de Moura ÉP, Dos Santos Maia M, Rodrigues GCS, de Medeiros HIR, Lopes SM, Scotti MT. Curr Neuropharmacol 20 857-885 (2022)
- Unveiling Natural and Semisynthetic Acylated Flavonoids: Chemistry and Biological Actions in the Context of Molecular Docking. El-Kersh DM, Abou El-Ezz RF, Fouad M, Farag MA. Molecules 27 5501 (2022)
Articles - 4bds mentioned but not cited (118)
- Functional constituents of wild and cultivated Goji (L. barbarum L.) leaves: phytochemical characterization, biological profile, and computational studies. Mocan A, Zengin G, Simirgiotis M, Schafberg M, Mollica A, Vodnar DC, Crişan G, Rohn S. J Enzyme Inhib Med Chem 32 153-168 (2017)
- A new crystal form of human acetylcholinesterase for exploratory room-temperature crystallography studies. Gerlits O, Ho KY, Cheng X, Blumenthal D, Taylor P, Kovalevsky A, Radić Z. Chem Biol Interact 309 108698 (2019)
- Sustainable Drug Discovery of Multi-Target-Directed Ligands for Alzheimer's Disease. Rossi M, Freschi M, de Camargo Nascente L, Salerno A, de Melo Viana Teixeira S, Nachon F, Chantegreil F, Soukup O, Prchal L, Malaguti M, Bergamini C, Bartolini M, Angeloni C, Hrelia S, Soares Romeiro LA, Bolognesi ML. J Med Chem 64 4972-4990 (2021)
- 7-Methoxytacrine-p-Anisidine Hybrids as Novel Dual Binding Site Acetylcholinesterase Inhibitors for Alzheimer's Disease Treatment. Korabecny J, Andrs M, Nepovimova E, Dolezal R, Babkova K, Horova A, Malinak D, Mezeiova E, Gorecki L, Sepsova V, Hrabinova M, Soukup O, Jun D, Kuca K. Molecules 20 22084-22101 (2015)
- DL0410 Ameliorates Memory and Cognitive Impairments Induced by Scopolamine via Increasing Cholinergic Neurotransmission in Mice. Lian W, Fang J, Xu L, Zhou W, Kang, Xiong W, Jia H, Liu AL, Du GH. Molecules 22 E410 (2017)
- Cholinesterase Inhibition Activity, Alkaloid Profiling and Molecular Docking of Chilean Rhodophiala (Amaryllidaceae). Tallini LR, Bastida J, Cortes N, Osorio EH, Theoduloz C, Schmeda-Hirschmann G. Molecules 23 E1532 (2018)
- Anti-Alzheimer potential, metabolomic profiling and molecular docking of green synthesized silver nanoparticles of Lampranthus coccineus and Malephora lutea aqueous extracts. Youssif KA, Haggag EG, Elshamy AM, Rabeh MA, Gabr NM, Seleem A, Salem MA, Hussein AS, Krischke M, Mueller MJ, Abdelmohsen UR. PLoS One 14 e0223781 (2019)
- Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer's disease therapy. Pachón-Angona I, Refouvelet B, Andrýs R, Martin H, Luzet V, Iriepa I, Moraleda I, Diez-Iriepa D, Oset-Gasque MJ, Marco-Contelles J, Musilek K, Ismaili L. J Enzyme Inhib Med Chem 34 479-489 (2019)
- Evaluation of neuroprotective and anti-amnesic effects of Elaeagnus umbellata Thunb. On scopolamine-induced memory impairment in mice. Nazir N, Zahoor M, Nisar M, Karim N, Latif A, Ahmad S, Uddin Z. BMC Complement Med Ther 20 143 (2020)
- Synthesis and Biological Evaluation of New Cholinesterase Inhibitors for Alzheimer's Disease. Hussein W, Sağlık BN, Levent S, Korkut B, Ilgın S, Özkay Y, Kaplancıklı ZA. Molecules 23 E2033 (2018)
- Antioxidant Molecules Isolated from Edible Prostrate Knotweed: Rational Derivatization to Produce More Potent Molecules. Mahnashi MH, Mahnashi MH, Alyami BA, Alqahtani YS, Alqarni AO, Jan MS, Hussain F, Zafar R, Rashid U, Abbas M, Tariq M, Sadiq A. Oxid Med Cell Longev 2022 3127480 (2022)
- Neuroprotective Potential of Synthetic Mono-Carbonyl Curcumin Analogs Assessed by Molecular Docking Studies. Hussain H, Ahmad S, Shah SWA, Ghias M, Ullah A, Rahman SU, Kamal Z, Khan FA, Khan NM, Muhammad J, Almehmadi M, Abdulaziz O, Alghamdi S. Molecules 26 7168 (2021)
- High-Throughput Screening and Molecular Dynamics Simulation of Natural Product-like Compounds against Alzheimer's Disease through Multitarget Approach. Iqbal D, Rehman MT, Bin Dukhyil A, Rizvi SMD, Al Ajmi MF, Alshehri BM, Banawas S, Khan MS, Alturaiki W, Alsaweed M. Pharmaceuticals (Basel) 14 937 (2021)
- Traditionally Used Lathyrus Species: Phytochemical Composition, Antioxidant Activity, Enzyme Inhibitory Properties, Cytotoxic Effects, and in silico Studies of L. czeczottianus and L. nissolia. Llorent-Martínez EJ, Zengin G, Fernández-de Córdova ML, Bender O, Atalay A, Ceylan R, Mollica A, Mocan A, Uysal S, Guler GO, Aktumsek A. Front Pharmacol 8 83 (2017)
- Novel N-allyl/propargyl tetrahydroquinolines: Synthesis via Three-component Cationic Imino Diels-Alder Reaction, Binding Prediction, and Evaluation as Cholinesterase Inhibitors. Rodríguez YA, Gutiérrez M, Ramírez D, Alzate-Morales J, Bernal CC, Güiza FM, Romero Bohórquez AR. Chem Biol Drug Des 88 498-510 (2016)
- Amaryllidaceae Alkaloids of Belladine-Type from Narcissus pseudonarcissus cv. Carlton as New Selective Inhibitors of Butyrylcholinesterase. Al Mamun A, Maříková J, Hulcová D, Janoušek J, Šafratová M, Nováková L, Kučera T, Hrabinová M, Kuneš J, Korábečný J, Cahlíková L. Biomolecules 10 E800 (2020)
- Combined in Vitro and in Silico Studies for the Anticholinesterase Activity and Pharmacokinetics of Coumarinyl Thiazoles and Oxadiazoles. Ibrar A, Khan A, Ali M, Sarwar R, Mehsud S, Farooq U, Halimi SMA, Khan I, Al-Harrasi A. Front Chem 6 61 (2018)
- Discovery of novel isoflavone derivatives as AChE/BuChE dual-targeted inhibitors: synthesis, biological evaluation and molecular modelling. Feng B, Li X, Xia J, Wu S. J Enzyme Inhib Med Chem 32 968-977 (2017)
- Exploring Structure-Activity Relationship in Tacrine-Squaramide Derivatives as Potent Cholinesterase Inhibitors. Svobodova B, Mezeiova E, Hepnarova V, Hrabinova M, Muckova L, Kobrlova T, Jun D, Soukup O, Jimeno ML, Marco-Contelles J, Korabecny J. Biomolecules 9 E379 (2019)
- Hippeastrum reticulatum (Amaryllidaceae): Alkaloid Profiling, Biological Activities and Molecular Docking. Tallini LR, Osorio EH, Santos VDD, Borges WS, Kaiser M, Viladomat F, Zuanazzi JAS, Bastida J. Molecules 22 E2191 (2017)
- Hydroxybenzoic Acid Derivatives as Dual-Target Ligands: Mitochondriotropic Antioxidants and Cholinesterase Inhibitors. Oliveira C, Cagide F, Teixeira J, Amorim R, Sequeira L, Mesiti F, Silva T, Garrido J, Remião F, Vilar S, Uriarte E, Oliveira PJ, Borges F. Front Chem 6 126 (2018)
- Attenuation of Scopolamine-Induced Amnesia via Cholinergic Modulation in Mice by Synthetic Curcumin Analogs. Hussain H, Ahmad S, Shah SWA, Ullah A, Ali N, Almehmadi M, Ahmad M, Khalil AAK, Jamal SB, Ahmad H, Halawi M. Molecules 27 2468 (2022)
- Microwave-Assisted Synthesis of (Piperidin-1-yl)quinolin-3-yl)methylene)hydrazinecarbothioamides as Potent Inhibitors of Cholinesterases: A Biochemical and In Silico Approach. Munir R, Zia-Ur-Rehman M, Murtaza S, Zaib S, Javid N, Awan SJ, Iftikhar K, Athar MM, Khan I. Molecules 26 656 (2021)
- Novel Tacrine-Scutellarin Hybrids as Multipotent Anti-Alzheimer's Agents: Design, Synthesis and Biological Evaluation. Spilovska K, Korabecny J, Sepsova V, Jun D, Hrabinova M, Jost P, Muckova L, Soukup O, Janockova J, Kucera T, Dolezal R, Mezeiova E, Kaping D, Kuca K. Molecules 22 E1006 (2017)
- Arylbenzofurans from the Root Bark of Morus alba as Triple Inhibitors of Cholinesterase, β-Site Amyloid Precursor Protein Cleaving Enzyme 1, and Glycogen Synthase Kinase-3β: Relevance to Alzheimer's Disease. Paudel P, Seong SH, Zhou Y, Ha MT, Min BS, Jung HA, Choi JS. ACS Omega 4 6283-6294 (2019)
- Derivatives of the β-Crinane Amaryllidaceae Alkaloid Haemanthamine as Multi-Target Directed Ligands for Alzheimer's Disease. Kohelová E, Peřinová R, Maafi N, Korábečný J, Hulcová D, Maříková J, Kučera T, Martínez González L, Hrabinova M, Vorčáková K, Nováková L, De Simone A, Havelek R, Cahlíková L. Molecules 24 E1307 (2019)
- Design and synthesis of multi-target directed 1,2,3-triazole-dimethylaminoacryloyl-chromenone derivatives with potential use in Alzheimer's disease. Karimi Askarani H, Iraji A, Rastegari A, Abbas Bukhari SN, Firuzi O, Akbarzadeh T, Saeedi M. BMC Chem 14 64 (2020)
- Identification of Compounds for Butyrylcholinesterase Inhibition. Li S, Li AJ, Travers J, Xu T, Sakamuru S, Klumpp-Thomas C, Huang R, Xia M. SLAS Discov 26 1355-1364 (2021)
- Analysis of Carotenoids in Haloarchaea Species from Atacama Saline Lakes by High Resolution UHPLC-Q-Orbitrap-Mass Spectrometry: Antioxidant Potential and Biological Effect on Cell Viability. Lizama C, Romero-Parra J, Andrade D, Riveros F, Bórquez J, Ahmed S, Venegas-Salas L, Cabalín C, Simirgiotis MJ. Antioxidants (Basel) 10 1230 (2021)
- Anti-Alzheimer's Disease Activity of Bromophenols from a Red Alga, Symphyocladia latiuscula (Harvey) Yamada. Paudel P, Seong SH, Zhou Y, Park HJ, Jung HA, Choi JS. ACS Omega 4 12259-12270 (2019)
- Discovery of novel choline acetyltransferase inhibitors using structure-based virtual screening. Kumar R, Kumar A, Långström B, Darreh-Shori T. Sci Rep 7 16287 (2017)
- Exploiting the Chalcone Scaffold to Develop Multifunctional Agents for Alzheimer's Disease. Rampa A, Bartolini M, Pruccoli L, Naldi M, Iriepa I, Moraleda I, Belluti F, Gobbi S, Tarozzi A, Bisi A. Molecules 23 (2018)
- In-Vitro, In-Vivo, Molecular Docking and ADMET Studies of 2-Substituted 3,7-Dihydroxy-4H-chromen-4-one for Oxidative Stress, Inflammation and Alzheimer's Disease. Mahnashi MH, Mahnashi MH, Alshahrani MA, Nahari MH, Hassan SSU, Jan MS, Ayaz M, Ullah F, Alshehri OM, Alshehri MA, Rashid U, Sadiq A. Metabolites 12 1055 (2022)
- Integration of in vitro and in silico perspectives to explain chemical characterization, biological potential and anticancer effects of Hypericum salsugineum: A pharmacologically active source for functional drug formulations. Bender O, Llorent-Martínez EJ, Zengin G, Mollica A, Ceylan R, Molina-García L, Fernández-de Córdova ML, Atalay A. PLoS One 13 e0197815 (2018)
- Multiple 3D-QSAR modeling, e-pharmacophore, molecular docking, and in vitro study to explore novel AChE inhibitors. Jana S, Ganeshpurkar A, Singh SK. RSC Adv 8 39477-39495 (2018)
- Synthesis and AChE-Inhibitory Activity of New Benzimidazole Derivatives. Acar Cevik U, Saglik BN, Levent S, Osmaniye D, Kaya Cavuşoglu B, Ozkay Y, Kaplancikli ZA. Molecules 24 E861 (2019)
- Synthesis of New Quinoline-Piperonal Hybrids as Potential Drugs against Alzheimer's Disease. de Oliveira C Brum J, Neto DCF, de Almeida JSFD, Lima JA, Kuca K, França TCC, Figueroa-Villar JD. Int J Mol Sci 20 E3944 (2019)
- Total Synthesis of Pulmonarin B and Design of Brominated Phenylacetic Acid/Tacrine Hybrids: Marine Pharmacophore Inspired Discovery of New ChE and Aβ Aggregation Inhibitors. Cheng ZQ, Song JL, Zhu K, Zhang J, Jiang CS, Zhang H. Mar Drugs 16 E293 (2018)
- Chemical Profiling and Cholinesterase Inhibitory Activity of Five Phaedranassa Herb. (Amaryllidaceae) Species from Ecuador. Moreno R, Tallini LR, Salazar C, Osorio EH, Montero E, Bastida J, Oleas NH, Acosta León K. Molecules 25 E2092 (2020)
- Design, Synthesis, and Bioevaluation of Indole Core Containing 2-Arylidine Derivatives of Thiazolopyrimidine as Multitarget Inhibitors of Cholinesterases and Monoamine Oxidase A/B for the Treatment of Alzheimer Disease. Shahid Nadeem M, Azam Khan J, Kazmi I, Rashid U. ACS Omega 7 9369-9379 (2022)
- Development of 2-Methoxyhuprine as Novel Lead for Alzheimer's Disease Therapy. Mezeiova E, Korabecny J, Sepsova V, Hrabinova M, Jost P, Muckova L, Kucera T, Dolezal R, Misik J, Spilovska K, Pham NL, Pokrievkova L, Roh J, Jun D, Soukup O, Kaping D, Kuca K. Molecules 22 E1265 (2017)
- Discovery of potent and selective butyrylcholinesterase inhibitors through the use of pharmacophore-based screening. Williams A, Zhou S, Zhan CG. Bioorg Med Chem Lett 29 126754 (2019)
- Multitarget Drug Design, Molecular Docking and PLIF Studies of Novel Tacrine-Coumarin Hybrids for the Treatment of Alzheimer's Disease. Fereidoonnezhad M, Mostoufi A, Eskandari M, Zali S, Aliyan F. Iran J Pharm Res 17 1217-1228 (2018)
- Neuroprotective derivatives of tacrine that target NMDA receptor and acetyl cholinesterase - Design, synthesis and biological evaluation. Remya C, Dileep KV, Koti Reddy E, Mantosh K, Lakshmi K, Sarah Jacob R, Sajith AM, Jayadevi Variyar E, Anwar S, Zhang KYJ, Sadasivan C, Omkumar RV. Comput Struct Biotechnol J 19 4517-4537 (2021)
- Rare genetic variability in human drug target genes modulates drug response and can guide precision medicine. Zhou Y, Arribas GH, Turku A, Jürgenson T, Mkrtchian S, Krebs K, Wang Y, Svobodova B, Milani L, Schulte G, Korabecny J, Gastaldello S, Lauschke VM. Sci Adv 7 eabi6856 (2021)
- Silibinin and Naringenin against Bisphenol A-Induced Neurotoxicity in Zebrafish Model-Potential Flavonoid Molecules for New Drug Design, Development, and Therapy for Neurological Disorders. Thayumanavan G, Jeyabalan S, Fuloria S, Sekar M, Ravi M, Selvaraj LK, Bala L, Chidambaram K, Gan SH, Rani NNIM, Begum MY, Subramaniyan V, Sathasivam KV, Meenakshi DU, Fuloria NK. Molecules 27 2572 (2022)
- Structure-Based Design and Discovery of a Long-Acting Cocaine Hydrolase Mutant with Improved Binding Affinity to Neonatal Fc Receptor for Treatment of Cocaine Abuse. Zheng F, Chen X, Kim K, Zhang T, Huang H, Zhou S, Zhang J, Jin Z, Zhan CG. AAPS J 22 62 (2020)
- Synthesis, in vitro screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivators. Malinak D, Dolezal R, Dolezal R, Hepnarova V, Hozova M, Andrys R, Bzonek P, Racakova V, Korabecny J, Gorecki L, Mezeiova E, Psotka M, Jun D, Kuca K, Musilek K. J Enzyme Inhib Med Chem 35 478-488 (2020)
- UHPLC-MS Metabolomic Fingerprinting, Antioxidant, and Enzyme Inhibition Activities of Himantormia lugubris from Antarctica. Areche C, Parra JR, Sepulveda B, García-Beltrán O, Simirgiotis MJ. Metabolites 12 560 (2022)
- Cholinesterase Inhibitory Activities of Adamantyl-Based Derivatives and Their Molecular Docking Studies. Kwong HC, Mah SH, Chia TS, Quah CK, Lim GK, Kumar CSC. Molecules 22 E1005 (2017)
- Comparative Evaluation of the Antioxidant and Anti-Alzheimer's Disease Potential of Coumestrol and Puerarol Isolated from Pueraria lobata Using Molecular Modeling Studies. Koirala P, Seong SH, Jung HA, Choi JS. Molecules 23 E785 (2018)
- Revealing the efficacy-toxicity relationship of Fuzi in treating rheumatoid arthritis by systems pharmacology. Feng W, Liu J, Zhang D, Tan Y, Cheng H, Peng C. Sci Rep 11 23083 (2021)
- The Distribution of Glucosinolates in Different Phenotypes of Lepidium peruvianum and Their Role as Acetyl- and Butyrylcholinesterase Inhibitors-In Silico and In Vitro Studies. Tarabasz D, Szczeblewski P, Laskowski T, Płaziński W, Baranowska-Wójcik E, Szwajgier D, Kukula-Koch W, Meissner HO. Int J Mol Sci 23 4858 (2022)
- 5-Methyl-N-(8-(5,6,7,8-tetrahydroacridin-9-ylamino)octyl)-5H-indolo[2,3-b]quinolin-11-amine: a highly potent human cholinesterase inhibitor. Wang L, Moraleda I, Iriepa I, Romero A, López-Muñoz F, Chioua M, Inokuchi T, Bartolini M, Marco-Contelles J. Medchemcomm 8 1307-1317 (2017)
- A Multidirectional Perspective for Novel Functional Products: In vitro Pharmacological Activities and In silico Studies on Ononis natrix subsp. hispanica. Yerlikaya S, Zengin G, Mollica A, Baloglu MC, Celik Altunoglu Y, Aktumsek A. Front Pharmacol 8 600 (2017)
- Alkaloids of Phaedranassa dubia (Kunth) J.F. Macbr. and Phaedranassa brevifolia Meerow (Amaryllidaceae) from Ecuador and its cholinesterase-inhibitory activity. León KA, Inca A, Tallini LR, Osorio EH, Robles J, Bastida J, Oleas NH. S Afr J Bot 136 91-99 (2021)
- Chromone-lipoic acid conjugate: Neuroprotective agent having acceptable butyrylcholinesterase inhibition, antioxidant and copper-chelation activities. Jalili-Baleh L, Nadri H, Forootanfar H, Küçükkılınç TT, Ayazgök B, Sharifzadeh M, Rahimifard M, Baeeri M, Abdollahi M, Foroumadi A, Khoobi M. Daru 29 23-38 (2021)
- Design, synthesis, and evaluation of novel cinnamic acid-tryptamine hybrid for inhibition of acetylcholinesterase and butyrylcholinesterase. Ghafary S, Ghobadian R, Mahdavi M, Nadri H, Moradi A, Akbarzadeh T, Najafi Z, Sharifzadeh M, Edraki N, Moghadam FH, Amini M. Daru 28 463-477 (2020)
- Exploring the Multi-Target Performance of Mitochondriotropic Antioxidants against the Pivotal Alzheimer's Disease Pathophysiological Hallmarks. Benfeito S, Fernandes C, Vilar S, Remião F, Uriarte E, Borges F. Molecules 25 E276 (2020)
- Metabolomic Profiling, Antioxidant and Enzyme Inhibition Properties and Molecular Docking Analysis of Antarctic Lichens. Torres-Benítez A, Ortega-Valencia JE, Sanchez M, Divakar PK, Simirgiotis MJ, Gómez-Serranillos MP. Molecules 27 8086 (2022)
- Molecular Dynamics Revealing a Detour-Forward Release Mechanism of Tacrine: Implication for the Specific Binding Characteristics in Butyrylcholinesterase. Zhang Z, Fan F, Luo W, Zhao Y, Wang C. Front Chem 8 730 (2020)
- New 1,2,3-Triazole-genipin Analogues and Their Anti-Alzheimer's Activity. Silalai P, Jaipea S, Tocharus J, Athipornchai A, Suksamrarn A, Saeeng R. ACS Omega 7 24302-24316 (2022)
- QuinoxalineTacrine QT78, a Cholinesterase Inhibitor as a Potential Ligand for Alzheimer's Disease Therapy. Ramos E, Palomino-Antolín A, Bartolini M, Iriepa I, Moraleda I, Diez-Iriepa D, Samadi A, Cortina CV, Chioua M, Egea J, Romero A, Marco-Contelles J. Molecules 24 E1503 (2019)
- Stephapierrines A-H, new tetrahydroprotoberberine and aporphine alkaloids from the tubers of Stephania pierrei Diels and their anti-cholinesterase activities. Chaichompoo W, Rojsitthisak P, Pabuprapap W, Siriwattanasathien Y, Yotmanee P, Haritakun W, Suksamrarn A. RSC Adv 11 21153-21169 (2021)
- Structure-based virtual screening leading to discovery of highly selective butyrylcholinesterase inhibitors with solanaceous alkaloid scaffolds. Zhou S, Yuan Y, Zheng F, Zhan CG. Chem Biol Interact 308 372-376 (2019)
- Succinimide Derivatives as Antioxidant Anticholinesterases, Anti-α-Amylase, and Anti-α-Glucosidase: In Vitro and In Silico Approaches. Alshehri OM, Mahnashi MH, Sadiq A, Zafar R, Jan MS, Ullah F, Alshehri MA, Alshamrani S, Hassan EE. Evid Based Complement Alternat Med 2022 6726438 (2022)
- UHPLC-MS Chemical Fingerprinting and Antioxidant, Antiproliferative, and Enzyme Inhibition Potential of Gaultheria pumila Berries. Fernández-Galleguillos C, Quesada-Romero L, Puerta A, Padrón JM, Souza E, Romero-Parra J, Simirgiotis MJ. Metabolites 11 523 (2021)
- Diclofenac derivatives as concomitant inhibitors of cholinesterase, monoamine oxidase, cyclooxygenase-2 and 5-lipoxygenase for the treatment of Alzheimer's disease: synthesis, pharmacology, toxicity and docking studies. Javed MA, Bibi S, Jan MS, Ikram M, Zaidi A, Farooq U, Sadiq A, Rashid U. RSC Adv 12 22503-22517 (2022)
- Discovery of Guanidine Derivatives from Buthus martensii Karsch with Metal-Binding and Cholinesterase Inhibition Properties. Liu YM, Fan JJ, Wang LN. Molecules 26 6737 (2021)
- Identification of a Novel Dual Inhibitor of Acetylcholinesterase and Butyrylcholinesterase: In Vitro and In Silico Studies. de Almeida RBM, Barbosa DB, do Bomfim MR, Amparo JAO, Andrade BS, Costa SL, Campos JM, Cruz JN, Santos CBR, Leite FHA, Botura MB. Pharmaceuticals (Basel) 16 95 (2023)
- Phenolic Profile, Antioxidant and Enzyme Inhibition Properties of the Chilean Endemic Plant Ovidia pillopillo (Gay) Meissner (Thymelaeaceae). Cortés C, González-Cabrera DA, Barrientos R, Parra C, Romero-Parra J, Pertino MW, Areche C, Sepúlveda B, Bórquez J, Torres-Benítez A, Simirgiotis MJ. Metabolites 12 90 (2022)
- Soyasapogenol-B as a Potential Multitarget Therapeutic Agent for Neurodegenerative Disorders: Molecular Docking and Dynamics Study. Iqbal D, Rizvi SMD, Rehman MT, Khan MS, Bin Dukhyil A, AlAjmi MF, Alshehri BM, Banawas S, Zia Q, Alsaweed M, Madkhali Y, Alsagaby SA, Alturaiki W. Entropy (Basel) 24 593 (2022)
- Structure Elucidation and Cholinesterase Inhibition Activity of Two New Minor Amaryllidaceae Alkaloids. Maříková J, Mamun AA, Shammari LA, Korábečný J, Kučera T, Hulcová D, Kuneš J, Malaník M, Vašková M, Kohelová E, Nováková L, Cahlíková L, Pour M. Molecules 26 1279 (2021)
- Synthesis, Biological Evaluation and Molecular Modelling of 2'-Hydroxychalcones as Acetylcholinesterase Inhibitors. Sukumaran SD, Chee CF, Viswanathan G, Buckle MJ, Othman R, Abd Rahman N, Chung LY. Molecules 21 E955 (2016)
- The insight of in vitro and in silico studies on cholinesterase inhibitors from the roots of Cimicifuga dahurica (Turcz.) Maxim. Kim JH, Thao NP, Han YK, Lee YS, Luyen BTT, Oanh HV, Kim YH, Yang SY. J Enzyme Inhib Med Chem 33 1174-1180 (2018)
- Chemical Composition, Antioxidant and Enzyme Inhibitory Activities of Onosma bourgaei and Onosma trachytricha and in Silico Molecular Docking Analysis of Dominant Compounds. Istifli ES. Molecules 26 2981 (2021)
- Cinnamomum verum J. Presl. Bark essential oil: in vitro investigation of anti-cholinesterase, anti-BACE1, and neuroprotective activity. Saeedi M, Iraji A, Vahedi-Mazdabadi Y, Alizadeh A, Edraki N, Firuzi O, Eftekhari M, Akbarzadeh T. BMC Complement Med Ther 22 303 (2022)
- Crystal Correlation Of Heterocyclic Imidazo[1,2-a]pyridine Analogues and Their Anticholinesterase Potential Evaluation. Kwong HC, Chidan Kumar CS, Mah SH, Mah YL, Chia TS, Quah CK, Lim GK, Chandraju S. Sci Rep 9 926 (2019)
- Design, Synthesis, and Biological Evaluation of a New Series of Biphenyl/Bibenzyl Derivatives Functioning as Dual Inhibitors of Acetylcholinesterase and Butyrylcholinesterase. Wang DM, Feng B, Fu H, Liu AL, Wang L, Du GH, Wu S. Molecules 22 E172 (2017)
- Design, synthesis, in silico and biological evaluations of novel polysubstituted pyrroles as selective acetylcholinesterase inhibitors against Alzheimer's disease. Pourtaher H, Hasaninejad A, Iraji A. Sci Rep 12 15236 (2022)
- Discovery of New Selective Butyrylcholinesterase (BChE) Inhibitors with Anti-Aβ Aggregation Activity: Structure-Based Virtual Screening, Hit Optimization and Biological Evaluation. Jiang CS, Ge YX, Cheng ZQ, Wang YY, Tao HR, Zhu K, Zhang H. Molecules 24 E2568 (2019)
- Engineering Dynamic Surface Peptide Networks on ButyrylcholinesteraseG117H for Enhanced Organophosphosphorus Anticholinesterase Catalysis. Hester KP, Bhattarai K, Jiang H, Agarwal PK, Pope C. Chem Res Toxicol 32 1801-1810 (2019)
- Is Caperatic Acid the Only Compound Responsible for Activity of Lichen Platismatia glauca within the Nervous System? Studzińska-Sroka E, Majchrzak-Celińska A, Bańdurska M, Rosiak N, Szwajgier D, Baranowska-Wójcik E, Szymański M, Gruszka W, Cielecka-Piontek J. Antioxidants (Basel) 11 2069 (2022)
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