Function and Biology

Crystal structure of BRD4 bromodomain 1 with N-methylpyrrolidin-2-one (NMP) derivative 18 (5-{[(3R)-1-methyl-5-oxopyrrolidin-3-yl]methyl}-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indol-1-one)

Source organism: Homo sapiens
Biochemical function: not assigned
Biological process: not assigned
Cellular component: not assigned

GO terms

Biochemical function:
  • not assigned
Biological process:
  • not assigned
Cellular component:
  • not assigned

Sequence family

Pfam Protein family (Pfam)
PF00439
Domain description: Bromodomain
Occurring in:
  1. Bromodomain-containing protein 4
The deposited structure of PDB entry 6psb contains 1 copy of Pfam domain PF00439 (Bromodomain) in Bromodomain-containing protein 4. Showing 1 copy in chain A.

InterPro InterPro annotations
IPR001487
Domain description: Bromodomain
Occurring in:
  1. Bromodomain-containing protein 4
IPR036427
Domain description: Bromodomain-like superfamily
Occurring in:
  1. Bromodomain-containing protein 4
IPR018359
Domain description: Bromodomain, conserved site
Occurring in:
  1. Bromodomain-containing protein 4
IPR043508
Domain description: Brdt, bromodomain, repeat I
Occurring in:
  1. Bromodomain-containing protein 4