Resolution: 3.9 Å
EM Method: Single-particle
Fitted PDBs: 8dn2
Q-score: 0.417
Nat Commun (2023) 14 pp. 6377-6377 [ DOI: doi:10.1038/s41467-023-42051-6 Pubmed: 37821459 ]
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Hexane (86 Da, Ligand)
- Decane (142 Da, Ligand)
- Heptane (100 Da, Ligand)
- Heteromeric glycine receptor subunit alpha-1 and beta, glycine-bound state 2(expanded-open state) (240 kDa, Complex from Homo sapiens)
- Undecane (156 Da, Ligand)
- N-octane (114 Da, Ligand)
- Glycine receptor subunit beta,green fluorescent protein,glycine receptor beta (76 kDa, Protein from Homo sapiens)
- N-butane (58 Da, Ligand)
- Glycine (75 Da, Ligand)
- Nonane (128 Da, Ligand)
- Glycine receptor subunit alpha-1 (42 kDa, Protein from Homo sapiens)
Cryo-EM structure of human Glycine Receptor alpha1-beta heteromer, apo state
Resolution: 3.55 Å
EM Method: Single-particle
Fitted PDBs: 8dn3
Q-score: 0.482
Nat Commun (2023) 14 pp. 6377-6377 [ DOI: doi:10.1038/s41467-023-42051-6 Pubmed: 37821459 ]
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Chloride ion (35 Da, Ligand)
- Heptane (100 Da, Ligand)
- Glycine receptor subunit beta,green fluorescent protein,glycine receptor beta (76 kDa, Protein from Homo sapiens)
- Hexane (86 Da, Ligand)
- Undecane (156 Da, Ligand)
- Glycine receptor subunit alpha-1 (42 kDa, Protein from Homo sapiens)
- Nonane (128 Da, Ligand)
- N-butane (58 Da, Ligand)
- Decane (142 Da, Ligand)
- Heteromeric glycine receptor alpha-1 and beta, apo state (240 kDa, Complex from Homo sapiens)
Resolution: 4.1 Å
EM Method: Single-particle
Fitted PDBs: 8dn4
Q-score: 0.373
Nat Commun (2023) 14 pp. 6377-6377 [ DOI: doi:10.1038/s41467-023-42051-6 Pubmed: 37821459 ]
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Heteromeric glycine receptor subunit alpha-1 and beta, glycine-bound state3(desensitized state) (240 kDa, Complex from Homo sapiens)
- Glycine receptor subunit beta,green fluorescent protein,glycine receptor beta (76 kDa, Protein from Homo sapiens)
- Hexane (86 Da, Ligand)
- Pentane (72 Da, Ligand)
- Glycine receptor subunit alpha-1 (42 kDa, Protein from Homo sapiens)
- Nonane (128 Da, Ligand)
- N-butane (58 Da, Ligand)
- N-octane (114 Da, Ligand)
Cryo-EM structure of human Glycine Receptor alpha1-beta heteromer, glycine-bound state1(open state)
Resolution: 3.63 Å
EM Method: Single-particle
Fitted PDBs: 8dn5
Q-score: 0.462
Nat Commun (2023) 14 pp. 6377-6377 [ DOI: doi:10.1038/s41467-023-42051-6 Pubmed: 37821459 ]
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Hexane (86 Da, Ligand)
- Decane (142 Da, Ligand)
- Heptane (100 Da, Ligand)
- Undecane (156 Da, Ligand)
- N-butane (58 Da, Ligand)
- Glycine receptor subunit beta,green fluorescent protein,glycine receptor beta (76 kDa, Protein from Homo sapiens)
- N-octane (114 Da, Ligand)
- Glycine (75 Da, Ligand)
- Nonane (128 Da, Ligand)
- Heteromeric glycine receptor subunit alpha-1 and beta, glycine-bound state1 (open state) (240 kDa, Complex from Homo sapiens)
- Glycine receptor subunit alpha-1 (42 kDa, Protein from Homo sapiens)
Resolution: 3.8 Å
EM Method: Single-particle
Fitted PDBs: 7sv7
Q-score: 0.463
Cell (2022) 185 pp. 158-168.e11 [ Pubmed: 34995514 DOI: doi:10.1016/j.cell.2021.12.009 ]
- Tetradecane (198 Da, Ligand)
- Adenosine-5'-triphosphate (507 Da, Ligand)
- Cystic fibrosis transmembrane conductance regulator (1 kDa, Protein from Homo sapiens)
- Dodecane (170 Da, Ligand)
- Cholesterol (386 Da, Ligand)
- Tezacaftor (520 Da, Ligand)
- Magnesium ion (24 Da, Ligand)
- Nonane (128 Da, Ligand)
- Cystic fibrosis transmembrane conductance regulator (168 kDa, Protein from Homo sapiens)
- The complex of phosphorylated human cystic fibrosis transmembrane conductance regulator (cftr) with atp/mg and tezacaftor (vx-661) (Complex from Homo sapiens)
- Heptadecane (240 Da, Ligand)
Resolution: 3.6 Å
EM Method: Single-particle
Fitted PDBs: 6x5b
Q-score: 0.396
Ozorowski G, Torres JL, Santos-Martins D, Forli S, Ward AB
Cell Rep (2020) 33 pp. 108428-108428 [ DOI: doi:10.1016/j.celrep.2020.108428 Pubmed: 33238117 ]
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- T-cell surface glycoprotein cd4 (23 kDa, Protein from Homo sapiens)
- Envelope glycoprotein gp120 (58 kDa, Protein from Human immunodeficiency virus 1)
- B41 hiv-1 env sosip in complex with soluble cd4, 17b fab, and small molecule go52 (630 kDa, Complex from Human immunodeficiency virus 1)
- Envelope glycoprotein gp41 (17 kDa, Protein from Human immunodeficiency virus 1)
- 17b fab heavy chain (24 kDa, Protein from Homo sapiens)
- 17b fab light chain (23 kDa, Protein from Homo sapiens)
- N-(4'-methyl[1,1'-biphenyl]-4-yl)-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide (336 Da, Ligand)
Resolution: 4.04 Å
EM Method: Single-particle
Fitted PDBs: 6x5c
Q-score: 0.341
Ozorowski G, Torres JL, Santos-Martins D, Forli S, Ward AB
Cell Rep (2020) 33 pp. 108428-108428 [ DOI: doi:10.1016/j.celrep.2020.108428 Pubmed: 33238117 ]
- B41 hiv-1 env sosip in complex with soluble cd4, 17b fab, and small molecule go52 (630 kDa, Complex from Human immunodeficiency virus 1)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Envelope glycoprotein gp41 (17 kDa, Protein from Human immunodeficiency virus 1)
- Envelope glycoprotein gp160 (58 kDa, Protein from Human immunodeficiency virus 1)
- N-(4'-methyl[1,1'-biphenyl]-4-yl)-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide (336 Da, Ligand)
- T-cell surface glycoprotein cd4 (23 kDa, Protein from Homo sapiens)
Human alpha3beta4 nicotinic acetylcholine receptor in complex with nicotine
Resolution: 3.34 Å
EM Method: Single-particle
Fitted PDBs: 6pv7
Q-score: 0.501
Gharpure A, Teng J, Zhuang Y, Noviello CM, Walsh Jr RM, Cabuco R, Howard RJ, Zaveri NT, Lindahl E, Hibbs RE
Neuron (2019) 104 pp. 501- [ DOI: doi:10.1016/j.neuron.2019.07.030 Pubmed: 31488329 ]
- Kappa fab light chain (23 kDa, Protein from house mouse)
- Igg2b heavy chain (Complex)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Human alpha3beta4 nicotinic acetylcholine receptor (Complex)
- Igg2b fab heavy chain (23 kDa, Protein from house mouse)
- Cholesterol hemisuccinate (486 Da, Ligand)
- (s)-3-(1-methylpyrrolidin-2-yl)pyridine (162 Da, Ligand)
- Neuronal acetylcholine receptor subunit beta-4 (Complex)
- Igg2b/kappa antibody (Complex)
- Nonane (128 Da, Ligand)
- Water (18 Da, Ligand)
- Fusion protein of neuronal acetylcholine receptor subunit alpha-3 and soluble cytochrome b562 (60 kDa, Protein from Homo sapiens)
- Human alpha3beta4 nicotinic receptor in complex with fab fragments and bound to nicotine (Complex from Homo sapiens)
- Neuronal acetylcholine receptor subunit alpha-3 (Complex)
- Kappa fab light chain (Complex)
- Fusion protein of neuronal acetylcholine receptor subunit beta-4 and soluble cytochrome b562 (61 kDa, Protein from Homo sapiens)
- Sodium ion (22 Da, Ligand)