EMD-23576
Structure of human 20S proteasome with bound MPI-5
EMD-23576
Single-particle3.4 Å
![EMD-23576](https://www.ebi.ac.uk/emdb/images/entry/EMD-23576/400_23576.gif)
Map released: 22/09/2021
Last modified: 13/04/2022
Sample Organism:
Human,
Plasmodium falciparum 3D7
Sample: Homo sapiens 20S proteasome complexed with ML052
Fitted models: 7lxv
Deposition Authors: Hanssen E
,
Xie SC
,
Liu B,
Leis AP,
Morton CJ
,
Metcalfe RD
,
Tilley L
,
Griffin MDW
Sample: Homo sapiens 20S proteasome complexed with ML052
Fitted models: 7lxv
Deposition Authors: Hanssen E
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Design of proteasome inhibitors with oral efficacy in vivo against Plasmodium falciparum and selectivity over the human proteasome.
Xie SC
,
Metcalfe RD
,
Mizutani H
,
Puhalovich T,
Hanssen E
,
Morton CJ
,
Du Y
,
Dogovski C,
Huang SC
,
Ciavarri J
,
Hales P
,
Griffin RJ
,
Cohen LH
,
Chuang BC,
Wittlin S,
Deni I
,
Yeo T
,
Ward KE
,
Barry DC
,
Liu B,
Gillett DL
,
Crespo-Fernandez BF
,
Ottilie S
,
Mittal N,
Churchyard A,
Ferguson D
,
Aguiar ACC
,
Guido RVC
,
Baum J
,
Hanson KK
,
Winzeler EA
,
Gamo FJ
,
Fidock DA
,
Baud D,
Parker MW
,
Brand S
,
Dick LR
,
Griffin MDW
,
Gould AE
,
Tilley L
(2021) PNAS , 118
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(2021) PNAS , 118