EMD-4590
Leishmania tarentolae proteasome 20S subunit complexed with GSK3494245
EMD-4590
Single-particle2.8 Å
![EMD-4590](https://www.ebi.ac.uk/emdb/images/entry/EMD-4590/400_4590.gif)
Map released: 17/04/2019
Last modified: 15/05/2024
Sample Organism:
Leishmania tarentolae
Sample: Proteasome 20S subunit
Fitted models: 6qm7
Deposition Authors: Rowland P, Goswami P
Sample: Proteasome 20S subunit
Fitted models: 6qm7
Deposition Authors: Rowland P, Goswami P
Preclinical candidate for the treatment of visceral leishmaniasis that acts through proteasome inhibition.
Wyllie S
,
Brand S
,
Thomas M,
De Rycker M
,
Chung CW,
Pena I,
Bingham RP,
Bueren-Calabuig JA,
Cantizani J,
Cebrian D,
Craggs PD
,
Ferguson L,
Goswami P,
Hobrath J,
Howe J,
Jeacock L,
Ko EJ
,
Korczynska J,
MacLean L,
Manthri S,
Martinez MS,
Mata-Cantero L,
Moniz S,
Nuhs A,
Osuna-Cabello M,
Pinto E,
Riley J,
Robinson S,
Rowland P,
Simeons FRC,
Shishikura Y,
Spinks D,
Stojanovski L,
Thomas J,
Thompson S,
Viayna Gaza E,
Wall RJ
,
Zuccotto F
,
Horn D
,
Ferguson MAJ,
Fairlamb AH
,
Fiandor JM,
Martin J,
Gray DW
,
Miles TJ,
Gilbert IH
,
Read KD,
Marco M
,
Wyatt PG
(2019) PNAS , 116 , 9318 - 9323
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(2019) PNAS , 116 , 9318 - 9323