Articles - 2dwo mentioned but not cited (3)
- IKKβ promotes metabolic adaptation to glutamine deprivation via phosphorylation and inhibition of PFKFB3. Reid MA, Lowman XH, Pan M, Tran TQ, Warmoes MO, Ishak Gabra MB, Yang Y, Locasale JW, Kong M. Genes Dev 30 1837-1851 (2016)
- Atroxlysin-III, A Metalloproteinase from the Venom of the Peruvian Pit Viper Snake Bothrops atrox (Jergón) Induces Glycoprotein VI Shedding and Impairs Platelet Function. Oliveira LS, Estevão-Costa MI, Alvarenga VG, Vivas-Ruiz DE, Yarleque A, Lima AM, Cavaco A, Eble JA, Sanchez EF. Molecules 24 E3489 (2019)
- Investigating combinatorial approaches in virtual screening on human inducible 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFKFB3): a case study for small molecule kinases. Crochet RB, Cavalier MC, Seo M, Kim JD, Yim YS, Park SJ, Lee YH. Anal Biochem 418 143-148 (2011)
Reviews citing this publication (2)
- Treatment against glucose-dependent cancers through metabolic PFKFB3 targeting of glycolytic flux. Jones BC, Pohlmann PR, Clarke R, Sengupta S. Cancer Metastasis Rev 41 447-458 (2022)
- Canonical and Non-Canonical Roles of PFKFB3 in Brain Tumors. Alvarez R, Mandal D, Chittiboina P. Cells 10 2913 (2021)
Articles citing this publication (8)
- Reduced methylation of PFKFB3 in cancer cells shunts glucose towards the pentose phosphate pathway. Yamamoto T, Takano N, Ishiwata K, Ohmura M, Nagahata Y, Matsuura T, Kamata A, Sakamoto K, Nakanishi T, Kubo A, Hishiki T, Suematsu M. Nat Commun 5 3480 (2014)
- Structure-based development of small molecule PFKFB3 inhibitors: a framework for potential cancer therapeutic agents targeting the Warburg effect. Seo M, Kim JD, Neau D, Sehgal I, Lee YH. PLoS One 6 e24179 (2011)
- Molecular basis of the fructose-2,6-bisphosphatase reaction of PFKFB3: transition state and the C-terminal function. Cavalier MC, Kim SG, Neau D, Lee YH. Proteins 80 1143-1153 (2012)
- Crystal structure of heart 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase (PFKFB2) and the inhibitory influence of citrate on substrate binding. Crochet RB, Kim JD, Lee H, Yim YS, Kim SG, Neau D, Lee YH. Proteins 85 117-124 (2017)
- Tuning PFKFB3 Bisphosphatase Activity Through Allosteric Interference. Macut H, Hu X, Tarantino D, Gilardoni E, Clerici F, Regazzoni L, Contini A, Pellegrino S, Luisa Gelmi M. Sci Rep 9 20333 (2019)
- Discovery and Structure-Activity Relationships of N-Aryl 6-Aminoquinoxalines as Potent PFKFB3 Kinase Inhibitors. Boutard N, Białas A, Sabiniarz A, Guzik P, Banaszak K, Biela A, Bień M, Buda A, Bugaj B, Cieluch E, Cierpich A, Dudek Ł, Eggenweiler HM, Fogt J, Gaik M, Gondela A, Jakubiec K, Jurzak M, Kitlińska A, Kowalczyk P, Kujawa M, Kwiecińska K, Leś M, Lindemann R, Maciuszek M, Mikulski M, Niedziejko P, Obara A, Pawlik H, Rzymski T, Sieprawska-Lupa M, Sowińska M, Szeremeta-Spisak J, Stachowicz A, Tomczyk MM, Wiklik K, Włoszczak Ł, Ziemiańska S, Zarębski A, Brzózka K, Nowak M, Fabritius CH. ChemMedChem 14 169-181 (2019)
- Structure-based design of small-molecule ligands of phosphofructokinase-2 activating or inhibiting glycolysis. Pyrkov TV, Sevostyanova IA, Schmalhausen EV, Shkoporov AN, Vinnik AA, Muronetz VI, Severin FF, Fedichev PO. ChemMedChem 8 1322-1329 (2013)
- Tumor chemical suffocation therapy by dual respiratory inhibitions. Xu Y, Guo Y, Chen L, Ni D, Hu P, Shi J. Chem Sci 12 7763-7769 (2021)