Structure analysis

BRAF in complex with an organic inhibitor 7898734

X-ray diffraction
2.55Å resolution
Source organism: Homo sapiens
Assemblies composition:
homo dimer
monomeric (preferred)
Entry contents: 1 distinct polypeptide molecule

Assemblies

Assembly 1
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Multimeric state: homo dimer
Accessible surface area: 24464.74 Å2
Buried surface area: 2195.6 Å2
Dissociation area: 1,097.8 Å2
Dissociation energy (ΔGdiss): -5.95 kcal/mol
Dissociation entropy (TΔSdiss): 13.38 kcal/mol
Symmetry number: 2
PDBe Complex ID: PDB-CPX-147199
Assembly 2 (preferred)
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Multimeric state: monomeric
Accessible surface area: 13629.63 Å2
Buried surface area: 0.0 Å2
Dissociation area: 0 Å2
Dissociation energy (ΔGdiss): 0 kcal/mol
Dissociation entropy (TΔSdiss): 0 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-147194
Assembly 3
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Multimeric state: monomeric
Accessible surface area: 13030.71 Å2
Buried surface area: 0.0 Å2
Dissociation area: 0 Å2
Dissociation energy (ΔGdiss): 0 kcal/mol
Dissociation entropy (TΔSdiss): 0 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-147194

Macromolecules

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