Structure analysis

PvSub1 Catalytic Domain in Complex with Peptidomimetic Inhibitor (MH-13)

X-ray diffraction
1.504Å resolution
Assembly composition:
hetero dimer (preferred)
Entry contents: 2 distinct polypeptide molecules

Assemblies

Assembly 1 (preferred)
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Multimeric state: hetero dimer
Accessible surface area: 13944.25 Å2
Buried surface area: 1702.63 Å2
Dissociation area: 593.29 Å2
Dissociation energy (ΔGdiss): -1.73 kcal/mol
Dissociation entropy (TΔSdiss): 6.1 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-241847
Assembly 2
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Multimeric state: hetero dimer
Accessible surface area: 14134.11 Å2
Buried surface area: 1460.08 Å2
Dissociation area: 555.6 Å2
Dissociation energy (ΔGdiss): -1 kcal/mol
Dissociation entropy (TΔSdiss): 6.08 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-241847

Macromolecules

Chains: A, B
Length: 631 amino acids
Theoretical weight: 69.89 KDa
Source organism: Plasmodium vivax
Expression system: Drosophila melanogaster
UniProt:
  • Canonical: E6Y8B9 (Residues: 26-630; Coverage: 100%)
Gene names: PVC01_100035100, PVT01_100029100, PVW1_100050600, sub1
Pfam:

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