GPR3 Orphan G-coupled Protein Receptor in complex with Dominant Negative Gs.
Resolution: 3.49 Å
EM Method: Single-particle
Fitted PDBs: 8u8f
Q-score: 0.422
Russell IC, Zhang X, Bumbak F, McNeill SM, Josephs TM, Leeming MG, Christopoulos G, Venugopal H, Flocco MM, Sexton PM, Wootten D, Belousoff MJ
Biochemistry (2024) 63 pp. 625-631 [ DOI: doi:10.1021/acs.biochem.3c00647 Pubmed: 38376112 ]
- Active state, gpr3 complex with dominant negative g-alphas. (Complex from Homo sapiens)
- Palmitic acid (256 Da, Ligand)
- Guanine nucleotide-binding protein g(i)/g(s)/g(o) subunit gamma-2 (6 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(i)/g(s)/g(t) subunit beta-1 (37 kDa, Protein from Homo sapiens)
- Guanine nucleotide-binding protein g(s) subunit alpha isoforms short (45 kDa, Protein from Homo sapiens)
- G-protein coupled receptor 3 (41 kDa, Protein from Homo sapiens)
Resolution: 2.9 Å
EM Method: Single-particle
Fitted PDBs: 6wqn
Q-score: 0.601
Wright A, Deane-Alder K, Marschall E, Bamert R, Venugopal H, Lithgow T, Lupton DW, Belousoff MJ
Acs Pharmacol Transl Sci (2020) 3 pp. 425-432 [ Pubmed: 32566908 DOI: doi:10.1021/acsptsci.0c00041 ]
- 50s ribosomal protein l2 (30 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l3 (23 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l28 (6 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l36 (4 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l24 (11 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l4 (22 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l29 (8 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l18 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l19 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal subunit (Complex from Staphylococcus aureus)
- 50s ribosomal protein l13 (16 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l16 (16 kDa, Protein from Staphylococcus aureus)
- 5s rrna (36 kDa, RNA from Staphylococcus aureus)
- 50s ribosomal protein l27 (9 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l21 (11 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l14 (13 kDa, Protein from Staphylococcus aureus)
- Contezolid (408 Da, Ligand)
- 50s ribosomal protein l15 (15 kDa, Protein from Staphylococcus aureus)
- 23s rrna (946 kDa, RNA from Staphylococcus aureus)
- 50s ribosomal protein l34 (6 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l22 (12 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l32 (6 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l23 (10 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l30 (6 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l20 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l33 (5 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l35 (7 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l25 (12 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l17 (13 kDa, Protein from Staphylococcus aureus)
Resolution: 3.1 Å
EM Method: Single-particle
Fitted PDBs: 6wqq
Q-score: 0.571
Wright A, Deane-Alder K, Marschall E, Bamert R, Venugopal H, Lithgow T, Lupton DW, Belousoff MJ
Acs Pharmacol Transl Sci (2020) 3 pp. 425-432 [ Pubmed: 32566908 DOI: doi:10.1021/acsptsci.0c00041 ]
- 50s ribosomal protein l20 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l18 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l16 (16 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l21 (11 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l30 (6 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l29 (8 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l14 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l36 (4 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l15 (15 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l4 (22 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l25 (12 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l13 (16 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l32 (6 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l22 (12 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l27 (9 kDa, Protein from Staphylococcus aureus)
- Radezolid (438 Da, Ligand)
- 50s ribosomal protein l23 (10 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l33 (5 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l17 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l3 (23 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l19 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal subunit (Complex from Staphylococcus aureus)
- 50s ribosomal protein l2 (30 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l24 (11 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l34 (6 kDa, Protein from Staphylococcus aureus)
- 23s rrna (946 kDa, RNA from Staphylococcus aureus)
- 50s ribosomal protein l35 (7 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l28 (6 kDa, Protein from Staphylococcus aureus)
- 5s rrna (36 kDa, RNA from Staphylococcus aureus)
Resolution: 3.2 Å
EM Method: Single-particle
Fitted PDBs: 6wrs
Q-score: 0.561
Wright A, Deane-Alder K, Marschall E, Bamert R, Venugopal H, Lithgow T, Lupton DW, Belousoff MJ
Acs Pharmacol Transl Sci (2020) 3 pp. 425-432 [ Pubmed: 32566908 DOI: doi:10.1021/acsptsci.0c00041 ]
- 50s ribosomal protein l2 (30 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l3 (23 kDa, Protein from Staphylococcus aureus)
- Ul22 (12 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l28 (6 kDa, Protein from Staphylococcus aureus)
- Tedizolid (370 Da, Ligand)
- 50s ribosomal protein l36 (4 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l24 (11 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l4 (22 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l29 (8 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l18 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l19 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal subunit (Complex from Staphylococcus aureus)
- 50s ribosomal protein l13 (16 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l16 (16 kDa, Protein from Staphylococcus aureus)
- 5s rrna (36 kDa, RNA from Staphylococcus aureus)
- 50s ribosomal protein l27 (9 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l21 (11 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l14 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l15 (15 kDa, Protein from Staphylococcus aureus)
- 23s rrna (946 kDa, RNA from Staphylococcus aureus)
- 50s ribosomal protein l34 (6 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l32 (6 kDa, Protein from Staphylococcus aureus)
- Ul25 (12 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l23 (10 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l30 (6 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l20 (13 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l33 (5 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l35 (7 kDa, Protein from Staphylococcus aureus)
- 50s ribosomal protein l17 (13 kDa, Protein from Staphylococcus aureus)